Acyl-CoA: cholesterol acyltransferase inhibitory activity of ginseng sapogenins, produced from the ginseng saponins

Bioorg Med Chem Lett. 1999 May 17;9(10):1375-8. doi: 10.1016/s0960-894x(99)00208-5.

Abstract

Ginseng sapogenins were produced from ginseng saponins, isolated from Korean ginseng roots. Ginseng saponins very mildly inhibited acyl-CoA:cholesterol acyltransferase (ACAT) in vitro, however, the sapogenins showed strong inhibitory activity on microsomal ACAT. Therefore, the sapogenins will be one of key ingredients of ginseng affected a lowering of the serum total cholesterol level.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anticholesteremic Agents / chemistry
  • Anticholesteremic Agents / isolation & purification
  • Anticholesteremic Agents / pharmacology
  • Enzyme Inhibitors / chemistry
  • Enzyme Inhibitors / isolation & purification
  • Enzyme Inhibitors / pharmacology*
  • Microsomes, Liver / drug effects
  • Microsomes, Liver / enzymology
  • Panax / chemistry*
  • Plants, Medicinal*
  • Rats
  • Sapogenins / chemistry
  • Sapogenins / isolation & purification
  • Sapogenins / pharmacology*
  • Saponins / chemistry*
  • Sterol O-Acyltransferase / antagonists & inhibitors*

Substances

  • Anticholesteremic Agents
  • Enzyme Inhibitors
  • Sapogenins
  • Saponins
  • Sterol O-Acyltransferase