Enzyme immunoassay detection of Cryptosporidium parvum inhibition by sinefungin in sporozoite infected HCT-8 enterocytic cells

Int J Parasitol. 1999 May;29(5):703-9. doi: 10.1016/s0020-7519(99)00031-4.

Abstract

Complete parasite development was obtained in differentiated human enterocytic HCT-8 cells infected at confluence with Cryptosporidium parvum sporozoites, and evaluated in a quantitative enzyme immunoassay. Forty-eight hours after infection, a linear correlation was found between optical density values and the number of parasites determined in an immunofluorescent assay. Sinefungin exerted an inhibitory effect when added within 4 h after sporozoite addition to HCT-8 cultures (MIC50 = 38 mumol L-1), while the inhibitory effects of paromomycin and pentamidine dimethanesulfonate were also easily detected (MIC50 = 0.87 mumol L-1 and 0.27 mumol L-1, respectively). Except for high pentamidine dimethanesulfonate concentrations, no alteration in optical microscopy morphology or trypan blue exclusion of HCT-8 cells was observed in the presence of anticryptosporidial agents, which suggests that they were primarily active against developing parasites. Data suggest that EIA detection of C. parvum development in sporozoite-infected HCT-8 cells provides an accurate and convenient model for in vitro evaluation of parasite infectivity, growth and response to anticryptosporidial agents.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine / analogs & derivatives*
  • Adenosine / pharmacology
  • Amebicides / pharmacology
  • Animals
  • Antiprotozoal Agents / pharmacology*
  • Cell Line
  • Cryptosporidium parvum / drug effects*
  • Cryptosporidium parvum / isolation & purification
  • Dose-Response Relationship, Drug
  • Fluorescent Antibody Technique, Indirect
  • Humans
  • Immunoenzyme Techniques / methods*
  • Parasite Egg Count
  • Paromomycin / pharmacology
  • Pentamidine / pharmacology
  • Rats
  • Rats, Sprague-Dawley
  • Time Factors

Substances

  • Amebicides
  • Antiprotozoal Agents
  • Paromomycin
  • Pentamidine
  • Adenosine
  • sinefungin