Disulfiram treatment for cocaine dependence in methadone-maintained opioid addicts

Addiction. 2000 Feb;95(2):219-28. doi: 10.1046/j.1360-0443.2000.9522198.x.

Abstract

Aims: Cocaine use by patients on methadone maintenance treatment is a widespread problem and is associated with a poorer prognosis. Recent studies have evaluated disulfiram as a treatment for individuals with comorbid alcohol and cocaine abuse. We evaluated the efficacy of disulfiram for cocaine dependence, both with and without co-morbid alcohol abuse, in a group of methadone-maintained opioid addicts.

Design: Randomized double-blind, placebo-controlled trial.

Setting: Urban methadone maintenance clinic.

Participants: Sixty-seven cocaine-dependent, methadone-maintained, opioid-dependent subjects (52% female; 51% Caucasian).

Intervention: Study medication, either disulfiram or placebo, was placed directly in the methadone to ensure compliance for 12 weeks.

Measurements: Primary outcome measures included weekly assessments of the frequency and quantity of drug and alcohol use, weekly urine toxicology screens and breathalyzer readings.

Findings: Disulfiram treated subjects decreased the quantity and frequency of cocaine use significantly more than those treated with placebo. Alcohol use was minimal for all subjects regardless of the medication.

Conclusions: Disulfiram may be an effective pharmacotherapy for cocaine abuse among methadone-maintained opioid addicts, even in those individuals without co-morbid alcohol abuse. Disulfiram inhibits dopamine beta-hydroxylase resulting in an excess of dopamine and decreased synthesis of norepinephrine. Since cocaine is a potent catecholamine re-uptake inhibitor, disulfiram may blunt cocaine craving or alter the "high", resulting in a decreased desire to use cocaine.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Cocaine-Related Disorders / complications
  • Cocaine-Related Disorders / drug therapy*
  • Disulfiram / therapeutic use*
  • Double-Blind Method
  • Enzyme Inhibitors / therapeutic use*
  • Female
  • Humans
  • Male
  • Methadone / therapeutic use
  • Narcotics / therapeutic use
  • Opioid-Related Disorders / complications*
  • Opioid-Related Disorders / rehabilitation

Substances

  • Enzyme Inhibitors
  • Narcotics
  • Disulfiram
  • Methadone