LMW-PTP exerts a differential regulation on PDGF- and insulin-mediated signaling

Biochem Biophys Res Commun. 2000 Apr 13;270(2):564-9. doi: 10.1006/bbrc.2000.2456.

Abstract

Low-molecular-weight protein tyrosine phosphatase (LMW-PTP) is able to specifically bind and dephosphorylate activated PDGF and insulin receptors, modulating the onset of mitogenic process. LMW-PTP is present in two distinct intracellular locations. While the cytosolic LMW-PTP pool interacts directly with activated insulin or PDGF receptors, the cytoskeleton-associated LMW-PTP is tyrosine phosphorylated upon PDGF stimulation and is involved in cytoskeleton rearrangement acting on p190Rho-GAP. We investigated the differential role of LMW-PTP in PDGF- or insulin-induced mitogenesis and cytoskeleton rearrangement. Dominant negative LMW-PTP influences both PDGF- and insulin-induced mitogenesis with a different extent and it induces a decrease in cellular adhesion and chemotaxis after PDGF but not insulin treatment. PDGF but not insulin stimulation leads to tyrosine phosphorylation of LMW-PTP. We propose that the differential effect of LMW-PTP on PDGF and insulin signaling is mainly due to the fact that during insulin signaling LMW-PTP does not become phosphorylated and thus does not act on its cytoskeleton-associated substrate/s.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Adhesion / drug effects
  • Cell Line
  • Chemotaxis / drug effects
  • Cytoskeleton / enzymology
  • Insulin / pharmacology*
  • Mice
  • Mitosis / drug effects
  • Molecular Weight
  • Phosphorylation
  • Platelet-Derived Growth Factor / pharmacology*
  • Protein Tyrosine Phosphatases / metabolism*
  • Signal Transduction / drug effects*
  • Tyrosine / metabolism

Substances

  • Insulin
  • Platelet-Derived Growth Factor
  • Tyrosine
  • Protein Tyrosine Phosphatases