Regional muramyl tripeptide phosphatidylethanolamine administration enhances hepatic immune function and tumor surveillance

Surgery. 2000 Aug;128(2):213-8. doi: 10.1067/msy.2000.107420.

Abstract

Background: Immune status of the liver may affect growth of liver metastases. We analyzed the ability of muramyl tripeptide phosphatidylethanolamine (MTP-PE), an immunomodulatory bacterial cell wall analog, to stimulate Kupffer cells (KCs) and protect against tumor growth, with or without an immunosuppressive partial hepatectomy (PH). Impact of MTP-PE's route of administration on KC function was assessed.

Methods: Buffalo rats (n = 7 to 12/group) were treated with saline, 40 microg MTP-PE intraportally (portal) or intravenously (IV) and challenged with 5 x 10(5) hepatoma cells, and tumors counted on day 21. To assess MTP-PE's impact on KC stimulation in animals undergoing PH, a known stimulant of tumor cell growth, groups were treated with saline or MTP-PE and challenged with tumor and underwent 30% PH. KCs were harvested and analyzed for superoxide production. Statistical analysis was performed with Mann-Whitney U test or chi-square test.

Results: MTP-PE-treated animals had fewer tumor nodules than control animals (19 vs 184, P <.005). MTP-PE-portal animals had fewer nodules than MTP-PE-IV (2 vs 36, P <.05). MTP-PE treatment before PH resulted in fewer tumor nodules compared with control animals (192 vs 276, P <. 05). MTP-PE administration increased macrophage superoxide production (20.6 +/- 2 vs 11.9 +/- 1.1 nmol/10(6) cells, P <.005).

Conclusions: MTP-PE improved KC function and decreased growth of microscopic tumor cells. MTP-PE's effects persist after an immunosuppressive hepatectomy. Portal administration was the most effective. MTP-PE administration may be useful as a neoadjuvant therapy for patients undergoing resection of liver malignancies.

MeSH terms

  • Acetylmuramyl-Alanyl-Isoglutamine / administration & dosage
  • Acetylmuramyl-Alanyl-Isoglutamine / analogs & derivatives*
  • Acetylmuramyl-Alanyl-Isoglutamine / pharmacology
  • Adjuvants, Immunologic / administration & dosage
  • Adjuvants, Immunologic / pharmacology*
  • Animals
  • Cell Division / drug effects
  • Drug Carriers
  • Hepatectomy
  • Infusions, Intravenous
  • Kupffer Cells / drug effects
  • Kupffer Cells / immunology*
  • Liposomes
  • Liver / drug effects
  • Liver / immunology
  • Liver Neoplasms, Experimental / immunology*
  • Liver Neoplasms, Experimental / pathology
  • Liver Neoplasms, Experimental / prevention & control
  • Phosphatidylethanolamines / administration & dosage
  • Phosphatidylethanolamines / pharmacology*
  • Portal System
  • Rats
  • Rats, Inbred BUF
  • Superoxides / metabolism

Substances

  • Adjuvants, Immunologic
  • Drug Carriers
  • Liposomes
  • Phosphatidylethanolamines
  • Superoxides
  • mifamurtide
  • Acetylmuramyl-Alanyl-Isoglutamine