Characterization of copper interactions with alzheimer amyloid beta peptides: identification of an attomolar-affinity copper binding site on amyloid beta1-42

J Neurochem. 2000 Sep;75(3):1219-33. doi: 10.1046/j.1471-4159.2000.0751219.x.

Abstract

Cu and Zn have been shown to accumulate in the brains of Alzheimer's disease patients. We have previously reported that Cu(2+) and Zn(2+) bind amyloid beta (Abeta), explaining their enrichment in plaque pathology. Here we detail the stoichiometries and binding affinities of multiple cooperative Cu(2+)-binding sites on synthetic Abeta1-40 and Abeta1-42. We have developed a ligand displacement technique (competitive metal capture analysis) that uses metal-chelator complexes to evaluate metal ion binding to Abeta, a notoriously self-aggregating peptide. This analysis indicated that there is a very-high-affinity Cu(2+)-binding site on Abeta1-42 (log K(app) = 17.2) that mediates peptide precipitation and that the tendency of this peptide to self-aggregate in aqueous solutions is due to the presence of trace Cu(2+) contamination (customarily approximately 0.1 microM). In contrast, Abeta1-40 has much lower affinity for Cu(2+) at this site (estimated log K(app) = 10.3), explaining why this peptide is less self-aggregating. The greater Cu(2+)-binding affinity of Abeta1-42 compared with Abeta1-40 is associated with significantly diminished negative cooperativity. The role of trace metal contamination in inducing Abeta precipitation was confirmed by the demonstration that Abeta peptide (10 microM) remained soluble for 5 days only in the presence of high-affinity Cu(2+)-selective chelators.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amyloid beta-Peptides / chemistry*
  • Amyloid beta-Peptides / metabolism*
  • Animals
  • Binding Sites
  • Chelating Agents / pharmacology
  • Copper / chemistry
  • Copper / metabolism*
  • Dogs
  • Humans
  • Kinetics
  • Peptide Fragments / chemistry*
  • Peptide Fragments / metabolism*
  • Regression Analysis
  • Serum Albumin / chemistry
  • Serum Albumin / metabolism
  • Zinc / metabolism

Substances

  • Amyloid beta-Peptides
  • Chelating Agents
  • Peptide Fragments
  • Serum Albumin
  • amyloid beta-protein (1-40)
  • amyloid beta-protein (1-42)
  • Copper
  • Zinc