Regulation of cardiac Jak-2 in animal models of insulin resistance

IUBMB Life. 2000 Jun;49(6):501-9. doi: 10.1080/15216540050167043.

Abstract

Insulin induces phosphorylation and activation of JAK2 tyrosine, as well as its association with STAT1 and SHP2 in insulin-sensitive tissues of intact rats, thus demonstrating a new pathway in transduction of insulin signals. We investigated this pathway in hearts of rats in three situations of insulin resistance: 72 h of fasting, chronic treatment with dexamethasone, and acute treatment with epinephrine. The acute treatment with epinephrine showed no difference in insulin-induced JAK2 tyrosine phosphorylation or JAK2/STAT1 and JAK2/SHP2 association in comparison with the control. In fasted rats the JAK2 protein concentration decreased, accompanied by a decrease in the stoichiometry of the phosphorylation to 70%, an increase in association of JAK2/STAT1 to 160%, and a decrease in JAK2/SHP2 association to 85%. In the dexamethasone-treated group, the JAK2 protein concentrations increased but the stoichiometry of its phosphorylation decreased to 20%, whereas the JAK2/STAT1 and JAK2/SHP2 associations changed by 70% and 170%, respectively. In fasting and dexamethasone-treated rats, therefore, insulin-induced JAK2 tyrosine phosphorylation decreases, and the JAK2 protein expression is differentially regulated such that the insulin-induced JAK2 association with SHP2 and STAT1 shows opposite interactions with the kinase.

MeSH terms

  • Animals
  • DNA-Binding Proteins / metabolism
  • Dexamethasone / pharmacology
  • Enzyme Activation / drug effects
  • Epinephrine / pharmacology
  • Fasting
  • Insulin Resistance / physiology*
  • Intracellular Signaling Peptides and Proteins
  • Janus Kinase 2
  • Male
  • Myocardium / enzymology*
  • Myocardium / metabolism
  • Phosphorylation
  • Protein Tyrosine Phosphatase, Non-Receptor Type 11
  • Protein Tyrosine Phosphatase, Non-Receptor Type 6
  • Protein Tyrosine Phosphatases / metabolism
  • Protein-Tyrosine Kinases / chemistry
  • Protein-Tyrosine Kinases / metabolism*
  • Proto-Oncogene Proteins*
  • Rats
  • Rats, Wistar
  • STAT1 Transcription Factor
  • Signal Transduction
  • Trans-Activators / metabolism
  • Tyrosine / metabolism

Substances

  • DNA-Binding Proteins
  • Intracellular Signaling Peptides and Proteins
  • Proto-Oncogene Proteins
  • STAT1 Transcription Factor
  • Stat1 protein, rat
  • Trans-Activators
  • Tyrosine
  • Dexamethasone
  • Protein-Tyrosine Kinases
  • Jak2 protein, rat
  • Janus Kinase 2
  • Protein Tyrosine Phosphatase, Non-Receptor Type 11
  • Protein Tyrosine Phosphatase, Non-Receptor Type 6
  • Protein Tyrosine Phosphatases
  • Ptpn11 protein, rat
  • Ptpn6 protein, rat
  • Epinephrine