Post-radiation severe xerostomia relieved by pilocarpine: a prospective French cooperative study

Radiother Oncol. 2000 Jun;55(3):233-9. doi: 10.1016/s0167-8140(99)00018-3.

Abstract

Background and purpose: The aim of the study was: (1) to confirm the action of pilocarpine hydrochloride (Salagen) against xerostomia: (2) to correlate the response to dose/volume radiotherapy parameters.

Materials and methods: From June 1995 to February 1996, 156 patients with severe radiation induced xerostomia received pilocarpine hydrochloride orally. IS mg per day with a 5 mg optional increase at S weeks up to a daily dose of 25 mg beyond 9 weeks.

Results: One hundred and forty five patients are fully evaluable. Treatment compliance was 75%. Thirty eight patients (26%) stopped treatment before week 12 for acute intolerance (sweating, nausea, vomiting) or no response. No severe complication occurred. Ninety ses en patients (67%) reported a significant relief of symptoms of xerostomia at 12 weeks. Within 12 weeks, the size of the subgroup ith normal food intake almost doubled (13-24 patients) while the size of the subgroup with (nearly) impossible solid food ingestion decreased by 38% (47 vs. 29 patients). The impact on quality of life was considered important or very important by 77% of the responders.

Conclusions: No difference was found according to dose/volume radiotherapy parameters suggesting that oral pilocarpine hydrochloride: (1) acts primarily by stimulating minor salivary glands: (2) can be of benefit to patients suffering of severe xerostomia regardless of radiotherapy dose/volume parameters: (3) all responders are identified at 12 weeks.

Publication types

  • Clinical Trial
  • Comparative Study
  • Randomized Controlled Trial

MeSH terms

  • Administration, Oral
  • Adult
  • Aged
  • Aged, 80 and over
  • Female
  • Head and Neck Neoplasms / radiotherapy
  • Humans
  • Male
  • Middle Aged
  • Muscarinic Agonists / administration & dosage
  • Muscarinic Agonists / therapeutic use*
  • Pilocarpine / administration & dosage
  • Pilocarpine / therapeutic use*
  • Prospective Studies
  • Quality of Life
  • Radiation Injuries / drug therapy*
  • Radiation Injuries / etiology
  • Radiotherapy / adverse effects
  • Saliva / metabolism
  • Salivary Glands / drug effects
  • Salivary Glands / metabolism
  • Salivary Glands / radiation effects*
  • Severity of Illness Index
  • Xerostomia / drug therapy*
  • Xerostomia / etiology

Substances

  • Muscarinic Agonists
  • Pilocarpine