Dopamine transporter density in young patients with schizophrenia assessed with [123]FP-CIT SPECT

Schizophr Res. 2001 Jan 15;47(1):59-67. doi: 10.1016/s0920-9964(00)00023-2.

Abstract

Disturbances in the dopamine (DA) system are thought to play a major role in schizophrenia. Amphetamine-induced release of endogenous DA is shown to be enhanced in schizophrenia, as is striatal [18F]FDOPA uptake in the striatum. It is not clear if the density of DA neurons is altered in schizophrenia. By studying the DA transporter with [123I]FP-CIT single photon emission computed tomography (SPECT), the density of nigrostriatal dopaminergic cells can be studied. Using [123I]FP-CIT SPECT, DA transporter density in the striatum was studied in 36 young patients with schizophrenia. Ten patients were antipsychotic (AP)-naive, 15 were treated with olanzapine, eight with risperidone and three were AP-free. A control group of 10 age-matched volunteers was included. Striatal [123I]FP-CIT binding was not significantly different between AP-naive patients (2.87), patients treated with olanzapine (2.76), patients treated with risperidone (2.76), AP-free patients (2.68) and controls (2.82) (F=0.07,p=0.98). Unexpectedly, striatal [123I]FP-CIT binding in females was significantly higher than in males (3.29 and 2.70, respectively; t=-2.56, p=0.014).Concluding, functional changes in the dopaminergic system in schizophrenia are not likely to be reflected in a change in DA transporter density. Moreover, DA transporter density does not seem to be altered by AP medication.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Benzodiazepines
  • Brain Mapping
  • Carrier Proteins / drug effects
  • Carrier Proteins / metabolism*
  • Corpus Striatum / diagnostic imaging
  • Corpus Striatum / drug effects
  • Dopamine Plasma Membrane Transport Proteins
  • Female
  • Humans
  • Iodine Radioisotopes
  • Male
  • Membrane Glycoproteins*
  • Membrane Transport Proteins*
  • Nerve Tissue Proteins*
  • Neural Pathways / diagnostic imaging
  • Neural Pathways / drug effects
  • Olanzapine
  • Pirenzepine / analogs & derivatives*
  • Pirenzepine / therapeutic use
  • Risperidone / therapeutic use
  • Schizophrenia / diagnostic imaging*
  • Schizophrenia / drug therapy
  • Substantia Nigra / diagnostic imaging
  • Substantia Nigra / drug effects
  • Tomography, Emission-Computed, Single-Photon*
  • Tropanes

Substances

  • Carrier Proteins
  • Dopamine Plasma Membrane Transport Proteins
  • Iodine Radioisotopes
  • Membrane Glycoproteins
  • Membrane Transport Proteins
  • Nerve Tissue Proteins
  • Tropanes
  • Benzodiazepines
  • 2-carbomethoxy-8-(3-fluoropropyl)-3-(4-iodophenyl)tropane
  • Pirenzepine
  • Risperidone
  • Olanzapine