New developments in the biology of the glucagon-like peptides GLP-1 and GLP-2

Ann N Y Acad Sci. 2000:921:226-32. doi: 10.1111/j.1749-6632.2000.tb06970.x.

Abstract

Glucagon-like peptides 1 and 2 (GLP-1 and GLP-2) are coencoded within a single mammalian proglucagon precursor, and are liberated in the intestine and brain. GLP-1 exerts well known actions on islet hormone secretion, gastric emptying, and food intake. Recent studies suggest GLP-1 plays a central role in the development and organization of islet cells. GLP-1 receptor signaling appears essential for beta cell signal transduction as exemplified by studies of GLP-1R-/- mice. GLP-2 promotes energy assimilation via trophic effects on the intestinal mucosa of the small and large bowel epithelium via a recently cloned GLP-2 receptor. The actions of GLP-2 are preserved in the setting of small and large bowel injury and inflammation. The biological actions of the glucagon-like peptides suggest they may have therapeutic efficacy in diabetes (GLP-1) or intestinal disorders (GLP-2).

Publication types

  • Review

MeSH terms

  • Animals
  • Diabetes Mellitus / therapy
  • Glucagon / physiology*
  • Glucagon-Like Peptide 1
  • Glucagon-Like Peptide 2
  • Glucagon-Like Peptide-1 Receptor
  • In Vitro Techniques
  • Intestinal Diseases / therapy
  • Intestinal Mucosa / physiology
  • Islets of Langerhans / growth & development
  • Islets of Langerhans / physiology
  • Mice
  • Mice, Knockout
  • Peptide Fragments / physiology*
  • Peptides / physiology*
  • Protein Precursors / physiology*
  • Receptors, Glucagon / genetics
  • Receptors, Glucagon / physiology
  • Signal Transduction

Substances

  • Glp1r protein, mouse
  • Glucagon-Like Peptide 2
  • Glucagon-Like Peptide-1 Receptor
  • Peptide Fragments
  • Peptides
  • Protein Precursors
  • Receptors, Glucagon
  • Glucagon-Like Peptide 1
  • Glucagon