Three key residues form a critical contact network in a protein folding transition state

Nature. 2001 Feb 1;409(6820):641-5. doi: 10.1038/35054591.

Abstract

Determining how a protein folds is a central problem in structural biology. The rate of folding of many proteins is determined by the transition state, so that a knowledge of its structure is essential for understanding the protein folding reaction. Here we use mutation measurements--which determine the role of individual residues in stabilizing the transition state--as restraints in a Monte Carlo sampling procedure to determine the ensemble of structures that make up the transition state. We apply this approach to the experimental data for the 98-residue protein acylphosphatase, and obtain a transition-state ensemble with the native-state topology and an average root-mean-square deviation of 6 A from the native structure. Although about 20 residues with small positional fluctuations form the structural core of this transition state, the native-like contact network of only three of these residues is sufficient to determine the overall fold of the protein. This result reveals how a nucleation mechanism involving a small number of key residues can lead to folding of a polypeptide chain to its unique native-state structure.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Acid Anhydride Hydrolases / chemistry*
  • Acid Anhydride Hydrolases / genetics
  • Acylphosphatase
  • Binding Sites
  • Models, Molecular
  • Monte Carlo Method
  • Mutation
  • Protein Conformation
  • Protein Folding*

Substances

  • Acid Anhydride Hydrolases