TEAD/TEF transcription factors utilize the activation domain of YAP65, a Src/Yes-associated protein localized in the cytoplasm

Genes Dev. 2001 May 15;15(10):1229-41. doi: 10.1101/gad.888601.

Abstract

Mammals express four highly conserved TEAD/TEF transcription factors that bind the same DNA sequence, but serve different functions during development. TEAD-2/TEF-4 protein purified from mouse cells was associated predominantly with a novel TEAD-binding domain at the amino terminus of YAP65, a powerful transcriptional coactivator. YAP65 interacted specifically with the carboxyl terminus of all four TEAD proteins. Both this interaction and sequence-specific DNA binding by TEAD were required for transcriptional activation in mouse cells. Expression of YAP in lymphocytic cells that normally do not support TEAD-dependent transcription (e.g., MPC11) resulted in up to 300-fold induction of TEAD activity. Conversely, TEAD overexpression squelched YAP activity. Therefore, the carboxy-terminal acidic activation domain in YAP is the transcriptional activation domain for TEAD transcription factors. However, whereas TEAD was concentrated in the nucleus, excess YAP65 accumulated in the cytoplasm as a complex with the cytoplasmic localization protein, 14-3-3. Because TEAD-dependent transcription was limited by YAP65, and YAP65 also binds Src/Yes protein tyrosine kinases, we propose that YAP65 regulates TEAD-dependent transcription in response to mitogenic signals.

MeSH terms

  • 3T3 Cells
  • Adaptor Proteins, Signal Transducing*
  • Animals
  • Carrier Proteins / metabolism*
  • Cell Cycle Proteins
  • Cytoplasm / metabolism*
  • DNA-Binding Proteins / chemistry
  • DNA-Binding Proteins / isolation & purification
  • DNA-Binding Proteins / metabolism*
  • Dimerization
  • Electrophoresis, Polyacrylamide Gel
  • Fluorescent Antibody Technique
  • Mass Spectrometry
  • Mice
  • Phosphoproteins / metabolism*
  • Protein Binding
  • Protein Structure, Tertiary
  • Subcellular Fractions / metabolism
  • TEA Domain Transcription Factors
  • Transcription Factors / chemistry
  • Transcription Factors / isolation & purification
  • Transcription Factors / metabolism*
  • Transcriptional Activation / genetics*
  • Transcriptional Activation / physiology
  • YAP-Signaling Proteins
  • src-Family Kinases / metabolism*

Substances

  • Adaptor Proteins, Signal Transducing
  • Carrier Proteins
  • Cell Cycle Proteins
  • DNA-Binding Proteins
  • Phosphoproteins
  • TEA Domain Transcription Factors
  • Tead2 protein, mouse
  • Transcription Factors
  • YAP-Signaling Proteins
  • Yap1 protein, mouse
  • src-Family Kinases