Abstract
Replacing the sugar-phosphodiester backbone of nucleic acids with a pyrrolidine-amide backbone results in an oligonucleotide mimic POM 1 which binds with high affinity and specificity to complementary DNA and RNA. Unlike other modified oligonucleotides, POM binds much more rapidly to single stranded RNA than DNA.
MeSH terms
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Amides / chemistry
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Amides / metabolism
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DNA / chemistry*
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DNA / metabolism
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Hydrogen-Ion Concentration
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Kinetics
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Molecular Mimicry
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Oligonucleotides / chemistry*
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Oligonucleotides / metabolism
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Osmolar Concentration
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Pyrrolidines / chemistry*
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Pyrrolidines / metabolism
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RNA / chemistry*
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RNA / metabolism
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Substrate Specificity
Substances
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Amides
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Oligonucleotides
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Pyrrolidines
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RNA
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DNA