Independent function of two destruction domains in hypoxia-inducible factor-alpha chains activated by prolyl hydroxylation

EMBO J. 2001 Sep 17;20(18):5197-206. doi: 10.1093/emboj/20.18.5197.

Abstract

Oxygen-dependent proteolytic destruction of hypoxia-inducible factor-alpha (HIF-alpha) subunits plays a central role in regulating transcriptional responses to hypoxia. Recent studies have defined a key function for the von Hippel-Lindau tumour suppressor E3 ubiquitin ligase (VHLE3) in this process, and have defined an interaction with HIF-1 alpha that is regulated by prolyl hydroxylation. Here we show that two independent regions within the HIF-alpha oxygen-dependent degradation domain (ODDD) are targeted for ubiquitylation by VHLE3 in a manner dependent upon prolyl hydroxylation. In a series of in vitro and in vivo assays, we demonstrate the independent and non-redundant operation of each site in regulation of the HIF system. Both sites contain a common core motif, but differ both in overall sequence and in the conditions under which they bind to the VHLE3 ligase complex. The definition of two independent destruction domains implicates a more complex system of pVHL-HIF-alpha interactions, but reinforces the role of prolyl hydroxylation as an oxygen-dependent destruction signal.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Motifs
  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Cattle
  • Cell Extracts / pharmacology
  • Conserved Sequence
  • Cytoplasm / physiology
  • DNA-Binding Proteins / chemistry*
  • DNA-Binding Proteins / metabolism*
  • Hydroxylation
  • Hypoxia-Inducible Factor 1
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Ligases*
  • Mice
  • Molecular Sequence Data
  • Nuclear Proteins / chemistry*
  • Nuclear Proteins / metabolism*
  • Proline / metabolism
  • Protein Structure, Tertiary
  • Proteins / physiology*
  • Sequence Homology, Amino Acid
  • Transcription Factors*
  • Tumor Suppressor Proteins*
  • Ubiquitin-Protein Ligases*
  • Ubiquitins / metabolism*
  • Von Hippel-Lindau Tumor Suppressor Protein

Substances

  • Cell Extracts
  • DNA-Binding Proteins
  • Hif1a protein, mouse
  • Hypoxia-Inducible Factor 1
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Nuclear Proteins
  • Proteins
  • Transcription Factors
  • Tumor Suppressor Proteins
  • Ubiquitins
  • Proline
  • Ubiquitin-Protein Ligases
  • Von Hippel-Lindau Tumor Suppressor Protein
  • Ligases