Phosphatidylinositol 3-kinase p85 adaptor function in T-cells. Co-stimulation and regulation of cytokine transcription independent of associated p110

J Biol Chem. 2002 Jan 11;277(2):912-21. doi: 10.1074/jbc.M107648200. Epub 2001 Oct 25.

Abstract

Phosphatidylinositol 3-kinase (PI3K) is a key regulator of a variety of cellular functions from cytoskeletal organization, vesicular trafficking, and cell proliferation to apoptosis. The enzyme complex is comprised of an 85-kDa adaptor (p85) coupled to a 110-kDa catalytic subunit (p110). While the function of PI3K has been largely attributed to the generation of D-3 lipids, an unanswered question has been whether p85 with a number of motifs (SH2, SH3, BcR homology (BH) region) can generate independent intracellular signals. In this study, we demonstrate that p85 lacking p110 (Deltap85) can activate NFAT transcription in T-cell hybridomas and normal splenocytes. This up-regulatory effect was unaffected by inhibition of PI 3-kinase, and cooperated specifically with Rac1, but not related family members. Stimulation correlated with Rac1 binding and was lost with the deletion of the BH domain. Lastly, the CD28-Deltap85 chimera also cooperated with TcR/CD3 to provide co-signals that enhanced IL-2 transcription. Our findings identify for the first time p85 as an adaptor that operates independently of the classic PI 3-kinase catalytic pathway and further shows that this pathway can provide co-signals in the regulation of T-cell function.

MeSH terms

  • Androstadienes / pharmacology
  • Animals
  • Cell Line
  • Cyclosporine / pharmacology
  • DNA-Binding Proteins / metabolism
  • Enzyme Inhibitors / pharmacology
  • Gene Expression Regulation*
  • Genes, Reporter
  • Humans
  • Hybridomas / physiology
  • Interleukin-2 / genetics*
  • Interleukin-2 / metabolism
  • Mice
  • NFATC Transcription Factors
  • Nuclear Proteins*
  • Phosphatidylinositol 3-Kinases / genetics
  • Phosphatidylinositol 3-Kinases / metabolism*
  • Promoter Regions, Genetic
  • Recombinant Fusion Proteins / metabolism
  • Signal Transduction*
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / enzymology
  • T-Lymphocytes / metabolism*
  • Transcription Factors / metabolism
  • Transcription, Genetic*
  • Up-Regulation
  • Wortmannin
  • rac1 GTP-Binding Protein / metabolism

Substances

  • Androstadienes
  • DNA-Binding Proteins
  • Enzyme Inhibitors
  • Interleukin-2
  • NFATC Transcription Factors
  • Nuclear Proteins
  • Recombinant Fusion Proteins
  • Transcription Factors
  • Cyclosporine
  • Phosphatidylinositol 3-Kinases
  • rac1 GTP-Binding Protein
  • Wortmannin