Sildenafil induces retinal vasodilatation in healthy subjects

Br J Ophthalmol. 2002 Feb;86(2):156-8. doi: 10.1136/bjo.86.2.156.

Abstract

Background: The cardiovascular effects of sildenafil (Viagra), a selective inhibitor of phosphodiesterase type 5 (PDE5), have been extensively studied. However, its effect on human retinal arteries and veins has not yet been investigated. The effect of a single dose administration of sildenafil on the retinal vessel diameters of healthy subjects was evaluated.

Methods: Sildenafil 50 mg was administered to 10 healthy subjects (male:female = 4:6; mean age 31 (SD 6) years). The diameters of retinal arteries and veins were measured by means of a retinal vessel analyser (RVA) immediately before and at 30, 60, 90, and 120 minutes after sildenafil uptake. Blood pressure, heart rate, and intraocular pressure were monitored in parallel.

Results: A significant increase of 5.8% (p<0.001) in both retinal arterial and venous diameters was found 30 minutes after sildenafil uptake. The diameters returned to baseline after 120 minutes. A mild systemic hypotensive response was seen. Changes in heart rate and intraocular pressure were not observed.

Conclusion: Sildenafil causes a significant dilatation of retinal arteries and veins in healthy subjects. A possible role for PDE5 in the regulation of retinal blood flow is implicated.

MeSH terms

  • Adult
  • Blood Pressure / drug effects
  • Female
  • Heart Rate / drug effects
  • Humans
  • Male
  • Nitric Oxide / physiology
  • Phosphodiesterase Inhibitors / adverse effects
  • Phosphodiesterase Inhibitors / pharmacology*
  • Piperazines / adverse effects
  • Piperazines / pharmacology*
  • Purines
  • Retinal Artery / drug effects
  • Retinal Artery / physiology
  • Retinal Vein / drug effects
  • Retinal Vein / physiology
  • Retinal Vessels / drug effects*
  • Sildenafil Citrate
  • Sulfones
  • Vasodilation / drug effects*

Substances

  • Phosphodiesterase Inhibitors
  • Piperazines
  • Purines
  • Sulfones
  • Nitric Oxide
  • Sildenafil Citrate