[In vitro activity of six fluoroquinolones and penicillin against 101 viridans group streptococci characterized by their susceptibility to erythromycin]

Rev Esp Quimioter. 2001 Dec;14(4):364-8.
[Article in Spanish]

Abstract

The increase in the use of the fluoroquinolones, including for the treatment of lower respiratory tract infections, seems to be associated with a parallel increase in bacterial resistance. We studied the activity of penicillin and six fluoroquinolones against 101 viridans group streptococci isolated from blood (58 erythromycin-susceptible and 43 erythromycin-resistant). The percentage of strains not susceptible to penicillin was 35% and there were statistically significant differences in the percentages of penicillin resistance between erythromycin-susceptible and -resistant strains. The fluoroquinolones studied showed good activity against our viridans group streptococci independent of their susceptibility to erythromycin. The norfloxacin MIC(50) and MIC(90) were 8 and 16 mg/l, respectively. Ofloxacin and ciprofloxacin showed the same activity (MIC(50) 1 mg/l and MIC(90) 2 mg/l); levofloxacin was similar with MIC(50) and MIC(90) of 1 mg/l. The fluoroquinolones with enhanced activity were moxifloxacin and trovafloxacin (MIC(50) 0.12 mg/l and MIC(90) 0.25 mg/l). However, we found two strains resistant to trovafloxacin (MIC = 4 mg/l) that showed reduced susceptibility to all the fluoroquinolones tested, including moxifloxacin (MIC = 2 mg/l). Mutations in the topoisomerase genes parC and gyrA have been shown to occur in strains with reduced susceptibility; therefore, ongoing surveillance for the development of fluoroquinolone resistance in viridans streptococci is necessary.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-Infective Agents / pharmacology*
  • Aza Compounds*
  • Bacteremia / microbiology
  • Ciprofloxacin / pharmacology
  • Drug Resistance
  • Drug Resistance, Multiple, Bacterial*
  • Erythromycin / pharmacology*
  • Fluoroquinolones*
  • Humans
  • Levofloxacin
  • Microbial Sensitivity Tests
  • Moxifloxacin
  • Naphthyridines / pharmacology
  • Norfloxacin / pharmacology
  • Ofloxacin / pharmacology
  • Penicillins / pharmacology*
  • Quinolines*
  • Streptococcal Infections / microbiology
  • Streptococcus / classification
  • Streptococcus / drug effects*
  • Streptococcus / isolation & purification

Substances

  • Anti-Infective Agents
  • Aza Compounds
  • Fluoroquinolones
  • Naphthyridines
  • Penicillins
  • Quinolines
  • Ciprofloxacin
  • Erythromycin
  • Levofloxacin
  • trovafloxacin
  • Ofloxacin
  • Norfloxacin
  • Moxifloxacin