Acute citalopram administration produces correlated increases in plasma and salivary cortisol

Psychopharmacology (Berl). 2002 Aug;163(1):118-20. doi: 10.1007/s00213-002-1149-4. Epub 2002 Jun 27.

Abstract

Rationale: Intravenous administration of the selective serotonin (5-HT) re-uptake inhibitor, citalopram, increases plasma cortisol. This would be expected to produce a parallel increase in salivary cortisol concentration.

Objective: To find out whether IV citalopram produces correlated increases in plasma and salivary cortisol levels.

Methods: Twelve healthy volunteers were tested on two occasions receiving either citalopram (10 mg IV) or saline in a double-blind, randomised, cross-over design. Plasma and salivary cortisol levels were measured before and for 150 min after each infusion.

Results: Relative to placebo, citalopram significantly increased cortisol levels in both plasma and saliva. The size of the increases in plasma and saliva cortisol correlated significantly with each other.

Conclusions: Monitoring changes in salivary cortisol might be a valid and acceptable means of measuring 5-HT-mediated cortisol release.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Area Under Curve
  • Citalopram / pharmacology*
  • Cross-Over Studies
  • Dose-Response Relationship, Drug
  • Double-Blind Method
  • Female
  • Humans
  • Hydrocortisone / blood
  • Hydrocortisone / metabolism*
  • Male
  • Middle Aged
  • Saliva / metabolism
  • Selective Serotonin Reuptake Inhibitors / pharmacology*

Substances

  • Serotonin Uptake Inhibitors
  • Citalopram
  • Hydrocortisone