Platelet glycoprotein IIb/IIIa receptor antagonist (abciximab) inhibited platelet activation and promoted skin flap survival after ischemia/reperfusion injury

J Surg Res. 2002 Sep;107(1):50-5. doi: 10.1006/jsre.2002.6500.

Abstract

Background: Evidence has shown that platelets play an important role in the pathogenesis of flap failure. Employing a rat inferior epigastric artery skin flap as a flap reperfusion injury model, we investigated whether platelet activation was involved in the skin flap failure and whether administration of abciximab (ReoPro, chimeric 7E3 Fab) could decrease platelet activation/aggregation and promote flap survival.

Methods: Normal saline and abciximab (0.06 mg/kg; 0.2 mg/kg; 1 mg/kg) were injected intravenously into skin flaps 30 min before reperfusion and 1 h after reperfusion (each subgroup n = 6). Platelet activation as demonstrated by P-selectin (CD62P) was analyzed by flow cytometry. P-selectin expression on flap vessels was detected by immunohistochemical staining. Platelet aggregation was induced with adenosine diphosphate (ADP). Laser Doppler flowmetry monitored tissue perfusion. The surviving area was evaluated 7 days postoperatively.

Results: CD62P progressively increased after reperfusion. The peak CD62P occurred after reperfusion for 12 h. Immunohistochemical staining showed CD62P significantly deposited on the endothelium after reperfusion. Administration of abciximab (1 mg/kg) effectively improved flap survival rate (P = 0.003), significantly decreased ADP-induced platelet aggregation (P < 0.001), and suppressed CD62P expression on blood platelets (P = 0.002) and its deposition on the flap vessels.

Conclusion: Abciximab promotion of skin flap survival is due to blocked platelet activation/aggregation and decreased activated-platelet deposition on the vascular endothelium. Thus, administration of a platelet glycoprotein IIb/IIIa receptor antagonist such as abciximab may save the skin flap from reperfusion injury after a long period of ischemia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Abciximab
  • Adenosine Diphosphate / pharmacology
  • Animals
  • Antibodies, Monoclonal / administration & dosage
  • Antibodies, Monoclonal / pharmacology*
  • Blood Platelets / drug effects
  • Blood Platelets / immunology
  • Dose-Response Relationship, Drug
  • Endothelium, Vascular / drug effects
  • Endothelium, Vascular / metabolism
  • Immunoglobulin Fab Fragments / administration & dosage
  • Immunoglobulin Fab Fragments / pharmacology*
  • Ischemia / physiopathology
  • Male
  • P-Selectin / metabolism
  • Platelet Activation / drug effects*
  • Platelet Aggregation / drug effects
  • Platelet Count
  • Platelet Glycoprotein GPIIb-IIIa Complex / antagonists & inhibitors*
  • Rats
  • Rats, Inbred Lew
  • Regional Blood Flow / drug effects
  • Reperfusion Injury / physiopathology
  • Skin / blood supply
  • Surgical Flaps / physiology*
  • Time Factors
  • Tissue Survival / drug effects*

Substances

  • Antibodies, Monoclonal
  • Immunoglobulin Fab Fragments
  • P-Selectin
  • Platelet Glycoprotein GPIIb-IIIa Complex
  • Adenosine Diphosphate
  • Abciximab