Past-A, a novel proton-associated sugar transporter, regulates glucose homeostasis in the brain

J Neurosci. 2002 Nov 1;22(21):9160-5. doi: 10.1523/JNEUROSCI.22-21-09160.2002.

Abstract

The ventral medullary surface (VMS) of the medulla oblongata is known to be the site of the central chemosensitive neurons in mammals. These neurons sense excess H+/CO2 dissolved in the CSF and induce hyperventilation. To elucidate the mechanism of neuronal cell adaptation to changes of H+/CO2, we screened for hypercapnia-induced genes in the VMS. Here, we report cloning and characterization of a novel gene called proton-associated sugar transporter-A (Past-A), which is induced in the brain after hypercapnia and mediates glucose uptake along the pH gradient. Past-A comprises 751 amino acid residues containing 12 membrane-spanning helices, several conserved sugar transport motifs, three proline-rich regions, and leucine repeats. Past-A transcript was expressed predominantly in the brain. Moreover, the Past-A-immunoreactive neural cells were found in the VMS of the medulla oblongata, and the number of immunoreactive cells was increased by hypercapnic stimulation. Transient transfection of Past-A in COS-7 cells leads to the expression of a membrane-associated 82 kDa protein that possesses a glucose transport activity. The acidification of extracellular medium facilitated glucose uptake, whereas the addition of carbonyl cyanide m-chlorophenylhydrazone, a protonophore, inhibited glucose import. Together, our results indicate that Past-A is a brain-specific glucose transporter that may represent an adaptation mechanism regulating sugar homeostasis in neuronal cells after hypercapnia.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Inhalation
  • Amino Acid Sequence
  • Animals
  • Biological Transport / physiology
  • Blotting, Northern
  • Brain / cytology
  • Brain / drug effects
  • Brain / metabolism*
  • COS Cells / metabolism
  • Carbon Dioxide / administration & dosage
  • Carrier Proteins / genetics
  • Carrier Proteins / metabolism*
  • Chemoreceptor Cells / drug effects
  • Chemoreceptor Cells / metabolism
  • Gene Expression Profiling
  • Glucose / metabolism*
  • Glucose / pharmacokinetics
  • Homeostasis / physiology*
  • Hydrogen-Ion Concentration
  • Hypercapnia / chemically induced
  • Hypercapnia / metabolism*
  • Immunohistochemistry
  • Male
  • Medulla Oblongata / cytology
  • Medulla Oblongata / drug effects
  • Medulla Oblongata / metabolism
  • Molecular Sequence Data
  • Monosaccharide Transport Proteins / genetics
  • Monosaccharide Transport Proteins / metabolism*
  • Neurons / drug effects
  • Neurons / metabolism
  • Organ Specificity
  • Phylogeny
  • Pons / cytology
  • Pons / drug effects
  • Pons / metabolism
  • RNA, Messenger / metabolism
  • Rats
  • Rats, Wistar

Substances

  • Carrier Proteins
  • Monosaccharide Transport Proteins
  • RNA, Messenger
  • Slc45a1 protein, rat
  • Carbon Dioxide
  • Glucose

Associated data

  • GENBANK/AB075229