[Antisense inhibition of cyclooxygenase-2 reduces malignant phenotype of gastric cancer cells]

Zhonghua Nei Ke Za Zhi. 2002 Aug;41(8):534-7.
[Article in Chinese]

Abstract

Objective: To investigate the role of cyclooxygenase-2 (COX-2) in tumorigenesis of gastric cancer, and the introduction of into human gastric cancer cells to suppress COX-2 expression.

Methods: The high COX-2 expressing human gastric cancer cell line SGC 7901 was stably transfected with the COX-2 antisense recombinant vector and plain vector (named as 7901-AS and 7901-P cells). The COX-2 expression levels in transfected cells were detected by immunocytochemistry and dot blotting methods. Proliferation and tumorigenic ability of transfected (7901-AS, 7901-P) and control (SGC 7901) cells were evaluated in vitro with MTT assay and in vivo with nude mice.

Results: Antisense treatment for COX-2 gene significantly reduced the expression level of COX-2 protein and mRNA and led inhibition of proliferation in 7901-AS cells. The tumor graft of 7901-AS in nude mice 30 days after implantation had less volume and weight than that of SGC7901 and 7901-P [(486.67 +/- 15.28) mg vs (826.67 +/- 77.67) mg and (776.67 +/- 300.06) mg, P < 0.01].

Conclusions: Overexpression of COX-2 in human gastric cancer cell line SGC 7901 was related to the malignant phenotype of cancer cells. Inhibition of COX-2 expression by antisense technique could reverse malignant phenotypes of gastric cancer cells.

Publication types

  • English Abstract

MeSH terms

  • Animals
  • Cell Division / genetics
  • Cell Division / physiology
  • Cyclooxygenase 2
  • DNA, Antisense / genetics*
  • DNA, Antisense / physiology
  • Gene Expression Regulation, Enzymologic
  • Humans
  • Immunohistochemistry
  • Isoenzymes / genetics*
  • Isoenzymes / metabolism
  • Membrane Proteins
  • Mice
  • Mice, Nude
  • Neoplasm Transplantation
  • Neoplasms, Experimental / enzymology
  • Neoplasms, Experimental / genetics
  • Neoplasms, Experimental / pathology
  • Phenotype
  • Prostaglandin-Endoperoxide Synthases / genetics*
  • Prostaglandin-Endoperoxide Synthases / metabolism
  • RNA, Messenger / genetics
  • RNA, Messenger / metabolism
  • Stomach Neoplasms / enzymology
  • Stomach Neoplasms / genetics
  • Stomach Neoplasms / pathology*
  • Tumor Cells, Cultured

Substances

  • DNA, Antisense
  • Isoenzymes
  • Membrane Proteins
  • RNA, Messenger
  • Cyclooxygenase 2
  • PTGS2 protein, human
  • Prostaglandin-Endoperoxide Synthases