Spatial and temporal aspects of Ca2+ signaling mediated by P2Y receptors in cultured rat hippocampal astrocytes

Life Sci. 2002 Dec 20;72(4-5):431-42. doi: 10.1016/s0024-3205(02)02273-7.

Abstract

ATP produces a variety of Ca2+ responses in astrocytes. To address the complex spatio-temporal Ca2+ signals, we analyzed the ATP-evoked increase in intracellular Ca2+ concentration ([Ca2+]i) in cultured rat hippocampal astrocytes using fura-2 or fluo-3 based Ca2+ imaging techniques. ATP at less than 10 nM produced elementary Ca2+ release event "puffs" in a manner independent of extracellular Ca2+. Stimulation with higher ATP concentrations (3 or 10 micro M) resulted in global Ca2+ responses such as intercellular Ca2+ wave. These Ca2+ responses were mainly mediated by metabotropic P2Y receptors. ATP acting on both P2Y1 and P2Y2 receptors produced a transient Ca2+ release by inositol 1,4,5-trisphosphate (InsP3). When cells were stimulated with ATP much longer, the transient [Ca2+]i elevation was followed by sustained Ca2+ entry from the extracellular space. This sustained rise in [Ca2+]i was inhibited by Zn2+ (<10 micro M), an inhibitor of capacitative Ca2+ entry (CCE). CCE induced by cyclopiazonic acid or thapsigargin and Ca2+ entry evoked by ATP share the same pharmacological profile in astrocytes. Taken together, the hierarchical Ca2+ responses to ATP were observed in hippocampal astrocytes, i.e., puffs, global Ca2+ release by InsP3, and CCE in response to depletion of InsP3-sensitive Ca2+ stores. It should be noted that these Ca2+ signals and their modulation by Zn2+ could occur in the hippocampus in situ since both ATP and Zn2+ are rich in the hippocampus and could be released by excitatory stimulation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / pharmacology
  • Animals
  • Astrocytes / drug effects*
  • Calcium / physiology
  • Calcium Channel Blockers / pharmacology
  • Calcium Signaling / drug effects*
  • Cations, Divalent / pharmacology
  • Cells, Cultured
  • Dose-Response Relationship, Drug
  • Enzyme Inhibitors / pharmacology
  • Hippocampus / cytology
  • Hippocampus / drug effects*
  • Indoles / pharmacology
  • Inositol 1,4,5-Trisphosphate / pharmacology
  • Microscopy, Confocal
  • Nicardipine / pharmacology
  • Rats
  • Rats, Wistar
  • Receptors, Purinergic / drug effects*
  • Uridine Triphosphate / pharmacology

Substances

  • Calcium Channel Blockers
  • Cations, Divalent
  • Enzyme Inhibitors
  • Indoles
  • Receptors, Purinergic
  • Inositol 1,4,5-Trisphosphate
  • Adenosine Triphosphate
  • Nicardipine
  • Calcium
  • Uridine Triphosphate
  • cyclopiazonic acid