R-Ras promotes focal adhesion formation through focal adhesion kinase and p130(Cas) by a novel mechanism that differs from integrins

Mol Cell Biol. 2003 Feb;23(3):933-49. doi: 10.1128/MCB.23.3.933-949.2003.

Abstract

R-Ras regulates integrin function, but its effects on integrin signaling pathways have not been well described. We demonstrate that activation of R-Ras promoted focal adhesion formation and altered localization of the alpha2beta1 integrin from cell-cell to cell-matrix adhesions in breast epithelial cells. Constitutively activated R-Ras(38V) dramatically enhanced focal adhesion kinase (FAK) and p130(Cas) phosphorylation upon collagen stimulation or clustering of the alpha2beta1 integrin, even in the absence of increased ligand binding. Signaling events downstream of R-Ras differed from integrins and K-Ras, since pharmacological inhibition of Src or disruption of actin inhibited integrin-mediated FAK and p130(Cas) phosphorylation, focal adhesion formation, and migration in control and K-Ras(12V)-expressing cells but had minimal effect in cells expressing R-Ras(38V). Therefore, signaling from R-Ras to FAK and p130(Cas) has a component that is Src independent and not through classic integrin signaling pathways and a component that is Src dependent. R-Ras effector domain mutants and pharmacological inhibition suggest a partial role for phosphatidylinositol 3-kinase (PI3K), but not Raf, in R-Ras signaling to FAK and p130(Cas). However, PI3K cannot account for the Src-independent pathway, since simultaneous inhibition of both PI3K and Src did not completely block effects of R-Ras on FAK phosphorylation. Our results suggest that R-Ras promotes focal adhesion formation by signaling to FAK and p130(Cas) through a novel mechanism that differs from but synergizes with the alpha2beta1 integrin.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Actins / metabolism
  • Cell Line
  • Collagen / metabolism
  • Crk-Associated Substrate Protein
  • Female
  • Focal Adhesion Kinase 1
  • Focal Adhesion Protein-Tyrosine Kinases
  • Focal Adhesions / physiology*
  • GTP Phosphohydrolases / chemistry
  • GTP Phosphohydrolases / physiology*
  • Humans
  • Integrin alpha2beta1 / physiology
  • Integrins / physiology*
  • Models, Biological
  • Phosphatidylinositol 3-Kinases / physiology
  • Phosphoproteins / physiology*
  • Phosphorylation
  • Protein Conformation
  • Protein-Tyrosine Kinases / physiology*
  • Proteins*
  • Proto-Oncogene Proteins pp60(c-src) / physiology
  • Retinoblastoma-Like Protein p130
  • Signal Transduction
  • ras Proteins / chemistry
  • ras Proteins / physiology*

Substances

  • Actins
  • BCAR1 protein, human
  • Crk-Associated Substrate Protein
  • Integrin alpha2beta1
  • Integrins
  • Phosphoproteins
  • Proteins
  • Retinoblastoma-Like Protein p130
  • Collagen
  • Phosphatidylinositol 3-Kinases
  • Protein-Tyrosine Kinases
  • Focal Adhesion Kinase 1
  • Focal Adhesion Protein-Tyrosine Kinases
  • PTK2 protein, human
  • Proto-Oncogene Proteins pp60(c-src)
  • GTP Phosphohydrolases
  • RRAS protein, human
  • ras Proteins