Prevalence and virologic consequences of HIV-1 genotype mutations detected in a cohort of 161 Italian patients receiving a nelfinavir-based highly active antiretroviral therapy

J Chemother. 2003 Apr;15(2):165-72. doi: 10.1179/joc.2003.15.2.165.

Abstract

A cross-sectional study was carried out in our tertiary care hospital between January 1998 and December 2001. All 161 consecutive patients naive to nelfinavir and who had received a nelfinavir-based highly active antiretroviral therapy (HAART) of at least 24-week duration were extrapolated from the 802 adult HIV-infected subjects treated with antiretroviral therapy. All cases of virologic failure were considered and viral genotyped. Virologic failure occurred in 80 out of 161 nelfinavir-treated patients, all belonging to the experienced group. On the whole, only 11 patients (7%) developed the D30N substitution, whose 6 was in association with the N88D mutation. Among the 80 failed patients, the M184V mutation was detected in 52 (65%), while only 7 patients showed simultaneously the M184V, T215Y and K103N substitutions. In our HIV-infected population receiving a nelfinavir-based HAART, the D30N mutation has shown a low absolute frequency, while the detection of M184V substitution and the simultaneous occurrence of M184V, T215Y and K103N mutations were related to a more favorable virological response.

MeSH terms

  • Adult
  • Antiretroviral Therapy, Highly Active*
  • Cross-Sectional Studies
  • DNA Mutational Analysis
  • DNA, Viral*
  • Drug Resistance, Viral / genetics*
  • Female
  • Genotype
  • HIV Infections / drug therapy*
  • HIV Protease Inhibitors / therapeutic use*
  • HIV-1 / genetics*
  • Humans
  • Italy
  • Male
  • Middle Aged
  • Nelfinavir / therapeutic use*
  • Prevalence
  • Treatment Outcome

Substances

  • DNA, Viral
  • HIV Protease Inhibitors
  • Nelfinavir