Stat6-protease but not Stat5-protease is inhibited by an elastase inhibitor ONO-5046

Biochem Biophys Res Commun. 2003 Oct 3;309(4):768-73. doi: 10.1016/j.bbrc.2003.08.067.

Abstract

A short isoform of Stat6 (65-kDa Stat6), a product of proteolytic processing by an undefined protease (Stat6-protease) in the nucleus, downregulates Stat6-mediated signaling in mast cells. Similarly, Stat5-mediated signaling is downregulated by Stat5-protease in myeloid progenitors. These proteases share a number of characteristics, including their nuclear localization and susceptibility to protease inhibitors. Here, we further investigated these Stat proteases. Interestingly, the activity of Stat6-protease but not of Stat5-protease was inhibited by ONO-5046, an elastase inhibitor that inhibits the activity of neutrophil elastase (NE) and NE-related protease proteinase 3 (PR3). Although both NE and PR3 were able to cleave Stat6 in vitro, the cleavage sites of Stat6 by NE or PR3 differed from that by Stat6-protease in mast cells. In addition, both NE and PR3 could also cleave Stat5, but they differed from Stat5-protease in myeloid progenitors. These results suggest that Stat6-protease may belong to the elastase family but differs from NE or PR3.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • DNA Primers
  • DNA-Binding Proteins / metabolism*
  • Enzyme Inhibitors / pharmacology*
  • Glycine / analogs & derivatives*
  • Glycine / pharmacology*
  • Mice
  • Mice, Inbred C57BL
  • Milk Proteins*
  • Pancreatic Elastase / antagonists & inhibitors*
  • Reverse Transcriptase Polymerase Chain Reaction
  • STAT5 Transcription Factor
  • STAT6 Transcription Factor
  • Sulfonamides / pharmacology*
  • Trans-Activators / antagonists & inhibitors*
  • Trans-Activators / metabolism*

Substances

  • DNA Primers
  • DNA-Binding Proteins
  • Enzyme Inhibitors
  • Milk Proteins
  • STAT5 Transcription Factor
  • STAT6 Transcription Factor
  • Stat6 protein, mouse
  • Sulfonamides
  • Trans-Activators
  • sivelestat
  • Pancreatic Elastase
  • Glycine