YM-14673, a new thyrotropin-releasing hormone analog, augments long-term potentiation in the mossy fiber-CA3 system of guinea pig hippocampal slices

J Pharmacobiodyn. 1992 Feb;15(2):75-8. doi: 10.1248/bpb1978.15.75.

Abstract

Effects of a new thyrotropin-releasing hormone (TRH) analog, N alpha-[[(S)-4-oxo-2-azetidinyl]carbonyl]L-histidyl-L-prolinamide dihydrate (YM-14673), which improves experimentally induced memory dysfunction, on long-term potentiation (LTP) in the mossy fiber-CA3 system, were investigated using guinea pig hippocampal slices. At concentrations of 10(-7) M and 10(-6) M, YM-14673 significantly augmented LTP in a concentration dependent manner. The magnitude of effect of 10(-6) M YM-14673 was similar to that of 10(-6) M TRH. As LTP in the hippocampus is regarded as an elementary process of memory and learning, the augmenting effect of YM-14673 on LTP in the present study may contribute to this drug's ability to remedy memory dysfunction.

MeSH terms

  • Animals
  • Azetidines / administration & dosage
  • Azetidines / pharmacology*
  • Dipeptides / administration & dosage
  • Dipeptides / pharmacology*
  • Dose-Response Relationship, Drug
  • Electric Stimulation
  • Electrophysiology
  • Guinea Pigs
  • Hippocampus / drug effects*
  • Hippocampus / physiology
  • Male
  • Nerve Fibers / drug effects*
  • Nerve Fibers / physiology
  • Thyrotropin-Releasing Hormone / analogs & derivatives

Substances

  • Azetidines
  • Dipeptides
  • Thyrotropin-Releasing Hormone
  • azetirelin