Cytological and ultrastructural investigation on osteoblastic and preosteoclastic cells grown in vitro in the presence of ipriflavone: preliminary results

Bone Miner. 1992 Oct:19 Suppl 1:S15-25. doi: 10.1016/0169-6009(92)90862-8.

Abstract

The effects of ipriflavone on bone cells were studied in vitro on pre-osteoclastic (FLG 29.1) and osteoblast-like (Saos-2) cells grown for 48 h either separately or in co-cultures, with or without the addition of PTH. Histological, ultrastructural and histochemical (TRAP-activity demonstration) methods were used. The main results show that ipriflavone reduces replication of FLG 29.1 cells and inhibits TRAP production by these cells both in controls and in co-cultures treated with PTH. Moreover, it has a moderate stimulatory effect on proliferation of osteoblast-like cells and reduces the PTH-induced degenerative changes of Saos-2 cells. These results suggest that the inhibitory effect of ipriflavone on FLG 29.1 cells might be indirect and might be mediated by the osteoblast-like cells.

MeSH terms

  • Acid Phosphatase / metabolism
  • Cell Adhesion / drug effects
  • Cell Division / drug effects
  • Filaggrin Proteins
  • Humans
  • Isoflavones / pharmacology*
  • Microscopy, Electron
  • Osteoblasts / drug effects*
  • Osteoblasts / ultrastructure
  • Osteoclasts / drug effects*
  • Osteoclasts / ultrastructure
  • Parathyroid Hormone / pharmacology
  • Tumor Cells, Cultured

Substances

  • FLG protein, human
  • Filaggrin Proteins
  • Isoflavones
  • Parathyroid Hormone
  • ipriflavone
  • Acid Phosphatase