Effectiveness of combined tamoxifen citrate and testosterone undecanoate treatment in men with idiopathic oligozoospermia

Fertil Steril. 2003 Oct;80(4):914-20. doi: 10.1016/s0015-0282(03)01123-3.

Abstract

Objective: To assess the effect of treatment with a combination of the antiestrogen tamoxifen citrate and the androgen testosterone undecanoate on sperm variables and pregnancy incidence in men with idiopathic oligozoospermia and couple subfertility.

Design: Prospective, randomized, placebo-controlled trial.

Setting: Clinical research in a tertiary care academic hospital.

Patient(s): Two hundred twelve men with idiopathic oligozoospermia and 82 normozoospermic men with female factor subfertility.

Intervention(s): Oligozoospermic patients were randomly assigned to two treatment groups with tamoxifen citrate, 20 mg/d, and testosterone undecanoate, 120 mg/d (n = 106) or placebo treatment (n = 106) for 6 months. Normozoospermic men were followed for the same period. Couple counseling was part of the intervention in all groups.

Main outcome measure(s): Pregnancy incidence and sperm characteristics after 3 and 6 months on medication and 3 months after the end of the trial.

Result(s): In the active treatment group, total sperm count (median [25th, 75th percentile], 27.1 x 10(6) cells/mL [9.4, 54.0 x 10(6) cells/mL] at baseline and 61.5 x 10(6) cells/mL [28.2, 119.6 x 10(6) cells/mL] at 6 months), progressive motility (mean [+/-SD], 29.7% +/- 12.0% at baseline and 41.6% +/- 13.1% at 6 months), and normal morphology (mean, 41.2% +/- 14.0% at baseline and 56.6% +/- 11.5% at 6 months) were noted. No marked changes were observed in placebo recipients or normozoospermic men. The incidence of spontaneous pregnancy was 33.9% in the active treatment group and 10.3% in the placebo group (36 vs. 11 pregnancies), with a relative risk of 3.195 (95% CI, 2.615 to 3.765).

Conclusion(s): Treatment with tamoxifen citrate and testosterone undecanoate improved sperm variables and led to a higher incidence of pregnancy in couples with subfertility related to idiopathic oligozoospermia.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Drug Therapy, Combination
  • Female
  • Humans
  • Male
  • Middle Aged
  • Oligospermia / drug therapy*
  • Placebos
  • Pregnancy
  • Pregnancy Rate
  • Risk
  • Sperm Count
  • Sperm Motility / drug effects
  • Spermatozoa / drug effects
  • Spermatozoa / physiology
  • Spermatozoa / ultrastructure
  • Tamoxifen / therapeutic use*
  • Testosterone / analogs & derivatives*
  • Testosterone / therapeutic use*
  • Testosterone Congeners / therapeutic use*

Substances

  • Placebos
  • Testosterone Congeners
  • Tamoxifen
  • Testosterone
  • testosterone undecanoate