Polypyrimidine tract-binding protein down-regulates fibroblast growth factor receptor 1 alpha-exon inclusion

Cancer Res. 2003 Oct 1;63(19):6154-7.

Abstract

Exclusion of the alpha-exon by alternative RNA splicing of the fibroblast growth factor receptor 1 (FGFR1) primary transcript leads to the production of FGFR1beta. Glial cell transformation is associated with a progressive increase in FGFR1beta expression that coincides with a dramatic increase in the expression of the splicing factor polypyrimidine tract-binding protein (PTB). Cell-specific overexpression of PTB increased alpha-exon skipping, and a reduction in PTB increased alpha-exon inclusion. Targeted disruption of PTB interaction with FGFR1 precursor RNA in vivo by an antisense oligonucleotide also increased alpha-exon inclusion. These results suggest that PTB plays a direct role in alpha-exon splicing.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alternative Splicing / drug effects
  • Alternative Splicing / genetics
  • Alternative Splicing / physiology*
  • Animals
  • Cell Line, Tumor
  • Down-Regulation
  • Exons / drug effects
  • Exons / genetics
  • Humans
  • Mice
  • Oligonucleotides, Antisense / genetics
  • Oligonucleotides, Antisense / pharmacology
  • Polypyrimidine Tract-Binding Protein / biosynthesis
  • Polypyrimidine Tract-Binding Protein / genetics
  • Polypyrimidine Tract-Binding Protein / physiology*
  • Protein Isoforms / biosynthesis
  • Protein Isoforms / genetics
  • RNA Precursors / drug effects
  • RNA Precursors / genetics
  • Receptor Protein-Tyrosine Kinases / biosynthesis
  • Receptor Protein-Tyrosine Kinases / genetics*
  • Receptor, Fibroblast Growth Factor, Type 1
  • Receptors, Fibroblast Growth Factor / biosynthesis
  • Receptors, Fibroblast Growth Factor / genetics*
  • Reverse Transcriptase Polymerase Chain Reaction

Substances

  • Oligonucleotides, Antisense
  • Protein Isoforms
  • RNA Precursors
  • Receptors, Fibroblast Growth Factor
  • Polypyrimidine Tract-Binding Protein
  • FGFR1 protein, human
  • Fgfr1 protein, mouse
  • Receptor Protein-Tyrosine Kinases
  • Receptor, Fibroblast Growth Factor, Type 1