Methylated hexitol nucleic acids, towards congeners with improved antisense potential

Nucleosides Nucleotides Nucleic Acids. 2003 May-Aug;22(5-8):1227-9. doi: 10.1081/NCN-120022842.

Abstract

In an effort to further improve the hybridisation potential of anhydro-hexitol nucleoside analogues, the 1'-methoxyl and 3'-methoxyl substituents were introduced and evaluated for their antisense potential. In view of the selectivity of pairing with RNA, especially the introduction of a 3'-O-alkyl moiety deserves further study.

MeSH terms

  • Alcohols*
  • Alkylation
  • Methylation
  • Nucleic Acids / chemical synthesis*
  • Nucleosides / chemical synthesis

Substances

  • Alcohols
  • Nucleic Acids
  • Nucleosides