Requirement of caspase-mediated cleavage of c-Abl during stress-induced apoptosis

Cell Death Differ. 2004 Mar;11(3):290-300. doi: 10.1038/sj.cdd.4401336.

Abstract

c-Abl protein tyrosine kinase plays an important role in cell cycle control and apoptosis. Furthermore, induction of apoptosis correlates with the activation of c-Abl. Here, we demonstrate the cleavage of c-Abl by caspases during apoptosis. Caspases separate c-Abl into functional domains including a Src-kinase, a fragment containing nuclear import sequences, a fragment with an actin-binding domain and nuclear export sequence. Caspase cleavage increases the kinase activity of c-Abl as demonstrated by in vitro kinase assays as well as by auto- and substrate phosphorylation. Cells in which c-Abl expression was knocked down by RNA interference resisted cisplatin- but not TNFalpha-induced apoptosis. A similar selective resistance against cisplatin-induced apoptosis was observed when cleavage resistant c-Abl was overexpressed in treated cells. Our data suggest the selective requirement of c-Abl cleavage by caspases for stress-induced, but not for TNFalpha-induced apoptosis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Motifs
  • Amino Acid Sequence
  • Animals
  • Antibodies, Monoclonal / metabolism
  • Apoptosis*
  • Blotting, Western
  • Caspases / metabolism*
  • Electrophoresis, Gel, Two-Dimensional
  • Electrophoresis, Polyacrylamide Gel
  • Enzyme Activation
  • Fluorescent Antibody Technique, Direct
  • HeLa Cells
  • Humans
  • Jurkat Cells
  • Mice
  • Microscopy, Confocal
  • Molecular Sequence Data
  • NIH 3T3 Cells
  • Polymerase Chain Reaction
  • Precipitin Tests
  • Protein Kinases / analysis
  • Protein Structure, Tertiary
  • Proto-Oncogene Proteins c-abl / chemistry
  • Proto-Oncogene Proteins c-abl / genetics
  • Proto-Oncogene Proteins c-abl / metabolism*
  • RNA Interference
  • Sequence Homology, Amino Acid
  • Stress, Physiological*
  • U937 Cells

Substances

  • Antibodies, Monoclonal
  • Protein Kinases
  • Proto-Oncogene Proteins c-abl
  • Caspases