Tramadol/acetaminophen combination tablets for the treatment of pain associated with osteoarthritis flare in an elderly patient population

J Am Geriatr Soc. 2004 Mar;52(3):374-80. doi: 10.1111/j.1532-5415.2004.52108.x.

Abstract

Objectives: To evaluate the efficacy and safety of adding tramadol 37.5 mg/acetaminophen (APAP) 325 mg combination tablets (tramadol/APAP) to existing therapy for painful osteoarthritis (OA) flare in a subset of elderly patients.

Design: Randomized, double-blind, placebo-controlled, 10-day add-on study.

Setting: Thirty outpatient centers.

Participants: Of 308 patients with painful OA flare, a subset of 113 patients aged 65 and older.

Measurements: Average daily pain intensity and pain relief scores for Days 1 through 5 and secondary quality-of-life measures and medication assessments.

Methods: Patients received one or two tramadol/APAP tablets or placebo four times per day for 10 days during ongoing nonselective or cyclooxygenase (COX)-2-selective nonsteroidal antiinflammatory drug (NSAID) therapy.

Results: Tramadol/APAP (n=69) was significantly superior to placebo (n=44) for average daily pain intensity (P=.034) and pain relief (P=.010) for Days 1 through 5 and Days 1 through 10 (P=.012 and P=.019, respectively). Tramadol/APAP had significantly better investigator (P<.001) and patient (P=.001) overall medication assessments and significantly better scores on three of four Western Ontario and McMaster Universities Osteoarthritis Index measures (P< or =.027). Most common adverse events with tramadol/APAP were nausea (18.8%), vomiting (13.0%), dizziness (11.6%), and constipation (4.3%), with an incidence similar to that of the overall study population. Mean daily dose of tramadol/APAP was 4.5 tablets (168 mg/1,458 mg).

Conclusion: Tramadol/APAP add-on therapy effectively managed painful OA flare in this elderly subset and was generally well tolerated.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetaminophen / administration & dosage*
  • Acetaminophen / adverse effects
  • Aged
  • Analgesics, Non-Narcotic / administration & dosage*
  • Analgesics, Non-Narcotic / adverse effects
  • Analgesics, Opioid / administration & dosage*
  • Analgesics, Opioid / adverse effects
  • Anti-Inflammatory Agents, Non-Steroidal / administration & dosage
  • Cyclooxygenase 2
  • Double-Blind Method
  • Drug Combinations
  • Female
  • Humans
  • Isoenzymes / administration & dosage
  • Male
  • Membrane Proteins
  • Osteoarthritis / drug therapy*
  • Pain / drug therapy
  • Prostaglandin-Endoperoxide Synthases / administration & dosage
  • Tablets
  • Tramadol / administration & dosage*
  • Tramadol / adverse effects

Substances

  • Analgesics, Non-Narcotic
  • Analgesics, Opioid
  • Anti-Inflammatory Agents, Non-Steroidal
  • Drug Combinations
  • Isoenzymes
  • Membrane Proteins
  • Tablets
  • Acetaminophen
  • Tramadol
  • Cyclooxygenase 2
  • PTGS2 protein, human
  • Prostaglandin-Endoperoxide Synthases