In the absence of type III receptor, the transforming growth factor (TGF)-beta type II-B receptor requires the type I receptor to bind TGF-beta2

J Biol Chem. 2004 May 21;279(21):22765-72. doi: 10.1074/jbc.M401350200. Epub 2004 Mar 2.

Abstract

Transforming growth factor beta (TGF-beta) ligands exert their biological effects through type II (TbetaRII) and type I receptors (TbetaRI). Unlike TGF-beta1 and -beta3, TGF-beta2 appears to require the co-receptor betaglycan (type III receptor, TbetaRIII) for high affinity binding and signaling. Recently, the TbetaRIII null mouse was generated and revealed significant non-overlapping phenotypes with the TGF-beta2 null mouse, implying the existence of TbetaRIII independent mechanisms for TGF-beta2 signaling. Because a variant of the type II receptor, the type II-B receptor (TbetaRII-B), has been suggested to mediate TGF-beta2 signaling in the absence of TbetaRIII, we directly tested the ability of TbetaRII-B to bind TGF-beta2. Here we show that the soluble extracellular domain of the type II-B receptor (sTbetaRII-B.Fc) bound TGF-beta1 and TGF-beta3 with high affinity (K(d) values = 31.7 +/- 22.8 and 74.6 +/- 15.8 pm, respectively), but TGF-beta2 binding was undetectable at corresponding doses. Similar results were obtained for the soluble type II receptor (sTbetaRII.Fc). However, sTbetaRII.Fc or sTbetaRII-B.Fc in combination with soluble type I receptor (sTbetaRI.Fc) formed a high affinity complex that bound TGF-beta2, and this complex inhibited TGF-beta2 in a biological inhibition assay. These results show that TGF-beta2 has the potential to signal in the absence of TbetaRIII when sufficient TGF-beta2, TbetaRI, and TbetaRII or TbetaRII-B are present. Our data also support a cooperative model for receptor-ligand interactions, as has been suggested by crystallization studies of TGF-beta receptors and ligands. Our cell-free binding assay system will allow for testing of models of receptor-ligand complexes prior to actual solution of crystal structures.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Activin Receptors, Type I / metabolism*
  • Animals
  • Blotting, Western
  • Cell Line
  • Cell Membrane / metabolism
  • Cell-Free System
  • Cloning, Molecular
  • Crystallography, X-Ray
  • DNA, Complementary / metabolism
  • Dose-Response Relationship, Drug
  • Genes, Reporter
  • Glycosylation
  • Humans
  • Kinetics
  • Ligands
  • Luciferases / metabolism
  • Mice
  • Models, Biological
  • Molecular Sequence Data
  • Phenotype
  • Protein Binding
  • Protein Isoforms
  • Protein Serine-Threonine Kinases
  • Protein Structure, Tertiary
  • Proteoglycans / metabolism*
  • Receptor, Transforming Growth Factor-beta Type I
  • Receptor, Transforming Growth Factor-beta Type II
  • Receptors, Transforming Growth Factor beta / metabolism*
  • Receptors, Transforming Growth Factor beta / physiology*
  • Signal Transduction

Substances

  • DNA, Complementary
  • Ligands
  • Protein Isoforms
  • Proteoglycans
  • Receptors, Transforming Growth Factor beta
  • betaglycan
  • Luciferases
  • Protein Serine-Threonine Kinases
  • Activin Receptors, Type I
  • Receptor, Transforming Growth Factor-beta Type I
  • Receptor, Transforming Growth Factor-beta Type II

Associated data

  • GENBANK/E10743