Abl-dependent tyrosine phosphorylation of Sos-1 mediates growth-factor-induced Rac activation

Nat Cell Biol. 2004 Mar;6(3):268-74. doi: 10.1038/ncb1096. Epub 2004 Feb 22.

Abstract

The non-receptor tyrosine kinase Abl participates in receptor tyrosine kinase (RTK)-induced actin cytoskeleton remodelling, a signalling pathway in which the function of Rac is pivotal. More importantly, the activity of Rac is indispensable for the leukaemogenic ability of the BCR-Abl oncoprotein. Thus, Rac might function downstream of Abl and be activated by it. Here, we elucidate the molecular mechanisms through which Abl signals to Rac in RTK-activated pathways. We show that Sos-1, a dual guanine nucleotide-exchange factor (GEF), is phosphorylated on tyrosine, after activation of RTKs, in an Abl-dependent manner. Sos-1 and Abl interact in vivo, and Abl-induced tyrosine phosphorylation of Sos-1 is sufficient to elicit its Rac-GEF activity in vitro. Genetic or pharmacological interference with Abl (and the related kinase Arg) resulted in a marked decrease in Rac activation induced by physiological doses of growth factors. Thus, our data identify the molecular connections of a pathway RTKs-Abl-Sos-1-Rac that is involved in signal transduction and actin remodelling.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Actin Cytoskeleton / enzymology*
  • Animals
  • COS Cells
  • Growth Substances / pharmacology
  • Humans
  • Phosphorylation / drug effects
  • Proto-Oncogene Proteins c-abl / antagonists & inhibitors
  • Proto-Oncogene Proteins c-abl / genetics
  • Proto-Oncogene Proteins c-abl / metabolism*
  • Receptor Protein-Tyrosine Kinases / drug effects
  • Receptor Protein-Tyrosine Kinases / metabolism*
  • SOS1 Protein / drug effects
  • SOS1 Protein / metabolism*
  • Signal Transduction / drug effects
  • Signal Transduction / physiology
  • Tyrosine / metabolism
  • rac GTP-Binding Proteins / drug effects
  • rac GTP-Binding Proteins / metabolism*

Substances

  • Growth Substances
  • SOS1 Protein
  • Tyrosine
  • Receptor Protein-Tyrosine Kinases
  • Proto-Oncogene Proteins c-abl
  • rac GTP-Binding Proteins