[Neuroprotective effects of topiramate]

Clin Ter. 2004 Feb-Mar;155(2-3):75-8.
[Article in Italian]

Abstract

Topiramate (TPM) is a new anti-convulsant drug, prescribed in epileptic seizure. Pharmacological actions of TPM are: a) a positive modulation of GABA receptors; b) inhibition of the kainite and aminohydroxymethylisoxazole propionic acid (AMPA) glutamate receptor sub-types; c) a use-dependent Na+ channel blocker. Recent studies suggest that TPM can have anti-excitotoxic properties, because it protects against motor neuron degeneration. Moreover, TPM enhances neuroprotection and reduces hemorrhagic incidence in focal cerebral ischemia.

Publication types

  • Review

MeSH terms

  • Anticonvulsants / pharmacology*
  • Anticonvulsants / therapeutic use
  • Fructose / analogs & derivatives*
  • Fructose / pharmacology*
  • Fructose / therapeutic use
  • Humans
  • Neuroprotective Agents / pharmacology*
  • Neuroprotective Agents / therapeutic use
  • Sodium Channels / drug effects
  • Topiramate
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid / antagonists & inhibitors

Substances

  • Anticonvulsants
  • Neuroprotective Agents
  • Sodium Channels
  • Topiramate
  • Fructose
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid