Characterization of a novel low-molecular-mass dual-specificity phosphatase-3 (LDP-3) that enhances activation of JNK and p38

Biochem J. 2004 Nov 1;383(Pt. 3):447-55. doi: 10.1042/BJ20040498.

Abstract

We have isolated a mouse cDNA for a novel dual-specificity phosphatase designated LDP-3 (low-molecular-mass dual-specificity phosphatase 3). The 450 bp open reading frame encodes a protein of 150 amino acids with a predicted molecular mass of 16 kDa. Northern blot and reverse transcription-PCR analyses show that LDP-3 transcripts are expressed in almost all mouse tissues examined. In vitro analyses using several substrates and inhibitors indicate that LDP-3 possesses intrinsic dual-specificity phosphatase activity. When expressed in mammalian cells, LDP-3 protein is localized mainly to the apical submembrane area. Forced expression of LDP-3 does not alter activation of ERK (extracellular-signal-regulated kinase), but rather enhances activation of JNK (c-Jun N-terminal kinase) and p38 and their respective upstream kinases MKK4 (mitogen-activated protein kinase kinase 4) and MKK6 in cells treated with 0.4 M sorbitol. By screening with a variety of stimuli, we found that LDP-3 specifically enhances the osmotic stress-induced activation of JNK and p38.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • COS Cells / enzymology
  • Cell Line
  • Chlorocebus aethiops
  • Dual-Specificity Phosphatases
  • Enzyme Activation / genetics
  • Enzyme Activation / physiology
  • Humans
  • JNK Mitogen-Activated Protein Kinases / metabolism*
  • MAP Kinase Kinase Kinase 4 / metabolism
  • Mice
  • Mitogen-Activated Protein Kinase 6 / metabolism
  • Molecular Sequence Data
  • Molecular Weight
  • Mutation / genetics
  • Mutation / physiology
  • Osmotic Pressure
  • Protein Tyrosine Phosphatases / chemistry*
  • Protein Tyrosine Phosphatases / genetics
  • Protein Tyrosine Phosphatases / physiology*
  • Substrate Specificity
  • Transfection / methods
  • p38 Mitogen-Activated Protein Kinases / metabolism*

Substances

  • JNK Mitogen-Activated Protein Kinases
  • Mitogen-Activated Protein Kinase 6
  • p38 Mitogen-Activated Protein Kinases
  • MAP Kinase Kinase Kinase 4
  • Dual-Specificity Phosphatases
  • Dusp23 protein, mouse
  • Protein Tyrosine Phosphatases

Associated data

  • GENBANK/AB164404
  • GENBANK/AB183013