Reconstitution and analysis of soluble inhibin and activin receptor complexes in a cell-free system

J Biol Chem. 2004 Dec 17;279(51):53126-35. doi: 10.1074/jbc.M408090200. Epub 2004 Oct 8.

Abstract

Activins and inhibins compose a heterogeneous subfamily within the transforming growth factor-beta (TGF-beta) superfamily of growth and differentiation factors with critical biological activities in embryos and adults. They signal through a heteromeric complex of type II, type I, and for inhibin, type III receptors. To characterize the affinity, specificity, and activity of these receptors (alone and in combination) for the inhibin/activin subfamily, we developed a cell-free assay system using soluble receptor-Fc fusion proteins. The soluble activin type II receptor (sActRII)-Fc fusion protein had a 7-fold higher affinity for activin A compared with sActRIIB-Fc, whereas both receptors had a marked preference for activin A over activin B. Although inhibin A and B binding was 20-fold lower compared with activin binding to either type II receptor alone, the mixture of either type II receptor with soluble TGF-beta type III receptor (TbetaRIII; betaglycan)-Fc reconstituted a soluble high affinity inhibin receptor. In contrast, mixing either soluble activin type II receptor with soluble activin type I receptors did not substantially enhance activin binding. Our results support a cooperative model of binding for the inhibin receptor (ActRII.sTbetaRIII complex) but not for activin receptors (type II + type I) and demonstrate that a complex composed of activin type II receptors and TbetaRIII is both necessary and sufficient for high affinity inhibin binding. This study also illustrates the utility of this cell-free system for investigating hypotheses of receptor complex mechanisms resulting from crystal structure analyses.

MeSH terms

  • Activin Receptors / chemistry*
  • Cell Line
  • Cell-Free System
  • Crystallography, X-Ray
  • Dose-Response Relationship, Drug
  • Electrophoresis, Polyacrylamide Gel
  • Glycosylation
  • Humans
  • Inhibins / chemistry*
  • Iodine / chemistry
  • Kinetics
  • Ligands
  • Protein Binding
  • Protein Structure, Tertiary
  • Receptors, Fc / chemistry
  • Recombinant Fusion Proteins / chemistry
  • Recombinant Fusion Proteins / metabolism
  • Recombinant Proteins / chemistry
  • Transforming Growth Factor beta / metabolism

Substances

  • Ligands
  • Receptors, Fc
  • Recombinant Fusion Proteins
  • Recombinant Proteins
  • Transforming Growth Factor beta
  • Inhibins
  • Iodine
  • Activin Receptors