Signal pathways in up-regulation of chemokines by tyrosine kinase MER/NYK in prostate cancer cells

Cancer Res. 2004 Oct 15;64(20):7311-20. doi: 10.1158/0008-5472.CAN-04-0972.

Abstract

The AXL/UFO family of tyrosine kinases is characterized by a common N-CAM (neural adhesion molecule)-related extracellular domain and a common ligand, GAS6 (growth arrest-specific protein 6). Family members are prone to transcriptional regulation and carry out diverse functions including the regulation of cell adhesion, migration, phagocytosis, and survival. In this report, we describe a new role of MER/N-CAM-related kinase (NYK), a member of the AXL family of kinases, in the up-regulation of chemokines in prostate cancer cells. We show that NYK has elevated expression in a subset of tumor specimens and prostate cancer cell lines. Activation of NYK in the prostate cancer cell line DU145 does not cause a mitogenic effect; instead, it causes a differentiation phenotype. Microarray analysis revealed that NYK is a strong inducer of endocrine factors including interleukin (IL)-8 and several other angiogenic CXC chemokines as well as bone morphogenic factors. The dramatic increase of IL-8 expression is seen at both transcriptional and posttranscriptional levels. The downstream signals engaged by NYK were characterized, and those responsible for the up-regulation of IL-8 transcription were defined. In contrast to IL-1alpha, NYK-induced up-regulation of IL-8 in DU145 depends on the mitogen-activated protein kinase kinase/extracellular signal-regulated kinase/Jun/Fos pathway, but not phosphoinositide 3'-kinase/nuclear factor-kappaB. These data define a new function of the AXL family of kinases and suggest a potential role of NYK in prostate cancer progression.

Publication types

  • Research Support, U.S. Gov't, Non-P.H.S.
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Base Sequence
  • Cell Line, Tumor
  • Enzyme Activation
  • Humans
  • Intercellular Signaling Peptides and Proteins / metabolism
  • Interleukin-8 / biosynthesis*
  • Interleukin-8 / genetics
  • MAP Kinase Signaling System / physiology
  • Male
  • Molecular Sequence Data
  • Promoter Regions, Genetic
  • Prostatic Neoplasms / enzymology
  • Prostatic Neoplasms / metabolism*
  • Protein Processing, Post-Translational
  • Proto-Oncogene Proteins / biosynthesis
  • Proto-Oncogene Proteins / metabolism*
  • Receptor Protein-Tyrosine Kinases / biosynthesis
  • Receptor Protein-Tyrosine Kinases / metabolism*
  • Transcriptional Activation
  • Up-Regulation
  • c-Mer Tyrosine Kinase

Substances

  • Intercellular Signaling Peptides and Proteins
  • Interleukin-8
  • Proto-Oncogene Proteins
  • growth arrest-specific protein 6
  • MERTK protein, human
  • Receptor Protein-Tyrosine Kinases
  • c-Mer Tyrosine Kinase