Conventional protein kinase C inhibition prevents alpha interferon-mediated hepatitis C virus replicon clearance by impairing STAT activation

J Virol. 2004 Dec;78(23):12809-16. doi: 10.1128/JVI.78.23.12809-12816.2004.

Abstract

Hepatitis C virus (HCV) has evolved complex strategies to evade host immune responses and establish chronic infection. The only treatment available for HCV infections, alpha interferon (IFN-alpha), is effective in a limited percentage of patients. The mechanisms by which IFN-alpha interferes with the HCV life cycle and the reasons for limited effectiveness of IFN-alpha therapy have not yet been fully elucidated. Using a cell-based HCV replication system and specific kinase inhibitors, we examined the role played by various signaling pathways in the IFN-alpha-mediated HCV clearance. We reported that conventional protein kinase C (cPKC) activity is important for the effectiveness of IFN-alpha treatment. In cells treated with a cPKC-specific inhibitor, IFN-alpha failed to induce an efficient HCV RNA degradation. The lack of cPKC activity leads to a broad reduction of IFN-alpha-stimulated gene expression due to a significant impairment of STAT1 and STAT3 tyrosine phosphorylation. Thus, modulation of cPKC function by either host or viral factors could influence the positive outcome of IFN-alpha-mediated antiviral therapies.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antiviral Agents / pharmacology*
  • Cell Line
  • DNA-Binding Proteins / metabolism*
  • Gene Expression Regulation, Viral / drug effects
  • Hepacivirus / drug effects*
  • Hepacivirus / genetics
  • Humans
  • Interferon-alpha / pharmacology*
  • Protein Kinase C / antagonists & inhibitors
  • Protein Kinase C / physiology*
  • RNA, Viral / metabolism
  • Replicon / drug effects*
  • STAT1 Transcription Factor
  • STAT3 Transcription Factor
  • Trans-Activators / metabolism*

Substances

  • Antiviral Agents
  • DNA-Binding Proteins
  • Interferon-alpha
  • RNA, Viral
  • STAT1 Transcription Factor
  • STAT1 protein, human
  • STAT3 Transcription Factor
  • STAT3 protein, human
  • Trans-Activators
  • Protein Kinase C