Transcriptional activation of integrin beta6 during the epithelial-mesenchymal transition defines a novel prognostic indicator of aggressive colon carcinoma

J Clin Invest. 2005 Feb;115(2):339-47. doi: 10.1172/JCI23183.

Abstract

We used a spheroid model of colon carcinoma to analyze integrin dynamics as a function of the epithelial-mesenchymal transition (EMT), a process that provides a paradigm for understanding how carcinoma cells acquire a more aggressive phenotype. This EMT involves transcriptional activation of the beta6 integrin subunit and a consequent induction of alphavbeta6 expression. This integrin enhances the tumorigenic properties of colon carcinoma, including activation of autocrine TGF-beta and migration on interstitial fibronectin. Importantly, this study validates the clinical relevance of the EMT. Kaplan-Meier analysis of beta6 expression in 488 colorectal carcinomas revealed a striking reduction in median survival time of patients with high beta6 expression. Elevated receptor expression did not simply reflect increasing tumor stage, since log-rank analysis showed a more significant impact on the survival of patients with early-stage, as opposed to late-stage, disease. Cox regression analysis confirmed that this integrin is an independent variable for these tumors. These findings define the alphavbeta6 integrin as an important risk factor for early-stage disease and a novel therapeutic candidate for colorectal cancer.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Autocrine Communication
  • Biomarkers, Tumor / biosynthesis*
  • Carcinoma / metabolism*
  • Carcinoma / pathology*
  • Colonic Neoplasms / metabolism*
  • Colonic Neoplasms / pathology*
  • Female
  • Gene Expression Regulation, Neoplastic
  • Humans
  • Integrin alpha5 / biosynthesis*
  • Integrin beta Chains / biosynthesis*
  • Intestinal Mucosa / pathology
  • Mesoderm / pathology
  • Mice
  • Mice, Nude
  • Neoplasm Invasiveness
  • Prognosis
  • Transcription, Genetic
  • Transforming Growth Factor beta / metabolism

Substances

  • Biomarkers, Tumor
  • Integrin alpha5
  • Integrin beta Chains
  • Transforming Growth Factor beta
  • integrin beta6