Low-dose terlipressin during long-term hyperdynamic porcine endotoxemia: effects on hepatosplanchnic perfusion, oxygen exchange, and metabolism

Crit Care Med. 2005 Feb;33(2):373-80. doi: 10.1097/01.ccm.0000152253.45901.fb.

Abstract

Objective: To investigate whether the vasopressin analog terlipressin might induce hepatosplanchnic ischemia during long-term, hyperdynamic, volume-resuscitated porcine endotoxemia.

Design: Prospective, randomized, controlled experimental study with repeated measures.

Setting: Investigational animal laboratory.

Subjects: Eighteen pigs were divided into two groups receiving either endotoxin alone (control group, n = 10) or endotoxin and terlipressin (n = 8).

Interventions: Pigs were anesthetized, mechanically ventilated, and instrumented and received a continuous intravenous infusion of Escherichia coli endotoxin. Animals were resuscitated with hydroxyethyl starch targeted to maintain mean arterial pressure >60 mm Hg. Twelve hours after the start of the endotoxin infusion, terlipressin (5-15 microg.kg.hr titrated to maintain mean arterial pressure at preendotoxin levels) or its vehicle was administered for 12 hrs.

Measurements and main results: Terlipressin increased mean arterial pressure and systemic vascular resistances, which was affiliated with a decrease in cardiac output and global oxygen consumption. Terlipressin restored the hepatic artery buffer response, which led to an increase in hepatic artery flow, ultimately resulting in well-maintained liver oxygen delivery, oxygen uptake, and all other variables of regional metabolism and organ function. Terlipressin markedly attenuated the hepatosplanchnic venous acidosis but was associated with pronounced hyperlactatemia.

Conclusions: During long-term hyperdynamic porcine endotoxemia, the well-known vasoconstrictor properties of terlipressin blunted the progressive decrease in mean arterial pressure without any detrimental effect on hepatosplanchnic perfusion, oxygen exchange, and metabolism. The marked terlipressin-induced hyperlactatemia did not originate from the hepatosplanchnic organs but from extrasplanchnic tissues, possibly muscle and skin.

Publication types

  • Research Support, Non-U.S. Gov't
  • Comment

MeSH terms

  • Animals
  • Blood Pressure / drug effects
  • Cardiac Output / drug effects
  • Endotoxemia / metabolism
  • Endotoxemia / physiopathology*
  • Endotoxins
  • Escherichia coli
  • Female
  • Glucose / metabolism
  • Hemodynamics / drug effects
  • Hydrogen-Ion Concentration
  • Lactic Acid / blood
  • Lipopolysaccharides
  • Liver Circulation / drug effects*
  • Lypressin / administration & dosage*
  • Lypressin / analogs & derivatives*
  • Male
  • Oxygen / blood
  • Oxygen Consumption / drug effects*
  • Pyruvic Acid / blood
  • Splanchnic Circulation / drug effects*
  • Swine
  • Terlipressin
  • Vascular Resistance / drug effects
  • Vasoconstrictor Agents / administration & dosage*

Substances

  • Endotoxins
  • Lipopolysaccharides
  • Vasoconstrictor Agents
  • Lactic Acid
  • Lypressin
  • endotoxin, Escherichia coli
  • Terlipressin
  • Pyruvic Acid
  • Glucose
  • Oxygen