Psychostimulants and G tolerance in rhesus monkeys: effects of oral modafinil and injected caffeine

Aviat Space Environ Med. 2005 Feb;76(2):121-6.

Abstract

Introduction: Caffeine and modafinil are psychostimulants that may be taken by fighter aircraft pilots to reduce fatigue. Fighter pilots are subjected to high positive G loads that reduce cerebral blood flow and consequently may induce G-LOC. The aim of the experiment was to determine whether these drugs may reduce tolerance to G stress.

Methods: Seven adult male rhesus monkeys participated in the experiment. Five were equipped with ECoG and ECG wires and underwent two G tests (A and B). Each experiment consisted of five centrifuge runs. Before the runs, the monkeys received no drug (control) or were given either 7.5 mg x kg(-1) caffeine IM or 64 mg x kg(-1) modafinil PO or the corresponding vehicles. The runs were performed up to +13 Gz with an onset rate of 0.1 G x s(-1) (test A) or 3 G x s(-1) (test B). The run was ended when the electrical activity of one ECoG channel had disappeared (i.e., G-LOC).

Results: In experiment A, drug administration had no significant effect. In experiment B, the injection of the caffeine-free solvent caused a delay in G-LOC compared with the control condition (no administration). Caffeine solvent also induced an increase in plasma osmolality.

Discussion: Modafinil administration has no significant effect on the G tolerance of rhesus monkeys. Regarding caffeine, the drug seems to have caused the reverse effect compared with the solvent.

Conclusions: Caffeine and modafinil administration had no significant effect on the G-tolerance of rhesus monkeys when compared with controls. This result needs to be confirmed in humans.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acceleration*
  • Aerospace Medicine
  • Animals
  • Benzhydryl Compounds / pharmacology*
  • Caffeine / pharmacology*
  • Central Nervous System Stimulants / pharmacology*
  • Centrifugation
  • Cerebral Cortex / drug effects
  • Cerebral Cortex / physiology
  • Electroencephalography
  • Electrooculography
  • Fatigue / etiology
  • Fatigue / prevention & control*
  • Hypergravity
  • Macaca mulatta
  • Male
  • Modafinil
  • Statistics, Nonparametric
  • Unconsciousness / etiology
  • Unconsciousness / prevention & control*

Substances

  • Benzhydryl Compounds
  • Central Nervous System Stimulants
  • Caffeine
  • Modafinil