[Regulation of orphan receptor ERR alpha by estrogen and progesterone in endometrial carcinoma cell line]

Beijing Da Xue Xue Bao Yi Xue Ban. 2005 Jun 18;37(3):281-3.
[Article in Chinese]

Abstract

Objective: To explore the relationship between expression of ERR alpha mRNA and estrogen and progesterone and to elucidate the function of ERR alpha in endometrial carcinoma.

Methods: The expression of ERR alpha mRNA was examined by reverse transcription polymerase chain reaction. Endometrial carcinoma cell line Ishikawa was dealt with different concentrations of 17beta-estradiol (10(-10) mol/L, 10(-8) mol/L and 10(-6) mol/L) for 15 min, 30 min and 24 h and 17beta-estradiol and ER inhibitor-ICI182780 were given concomitantly to observe the change of ERR alpha mRNA. Different concentrations of progesterone (10(-8) mol/L, 10(-7) mol/L, 10(-6) mol/L and 10(-5) mol/L) were also given to Ishikawa cell line for 24 h to observe the change of ERR alpha mRNA.

Results: The expression level of ERR alpha mRNA was slightly higher than that of the control group after being stimulated for 15 min, 30 min and 24 h by 10(-10) mol/L 17beta-estradiol. However the expression level of ERR alpha mRNA was significantly lower than that of the control group after being stimulated for 15 min, 30 min and 24 h by 10(-8) mol/L and 10(-6) mol/L of 17beta-estradiol. When 10(-6) mol/L of ICI182780 and 10(-8) mol/L of 17beta-estradiol were given simultaneously to Ishikawa cell line, this down-regulation was blocked. After being stimulated for 24 h by 10(-7) mol/L, 10(-6) mol/L and 10(-5) mol/L of progesterone, the expression levels of ERR alpha mRNA were significantly higher than that of the control group, but no change was found in 10(-8) mol/L of progesterone.

Conclusion: 17Beta-estradiol can down-regulate the expression of ERR alpha mRNA and this regulation is mediated by estrogen receptor. Progesterone can up-regulate the expression of ERR alpha mRNA.

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line, Tumor
  • Endometrial Neoplasms / metabolism*
  • Estradiol / pharmacology*
  • Female
  • Humans
  • Progesterone / pharmacology*
  • RNA, Messenger / biosynthesis
  • Receptors, Estrogen / biosynthesis*
  • Receptors, Estrogen / genetics
  • Reverse Transcriptase Polymerase Chain Reaction
  • Uterine Neoplasms / metabolism*

Substances

  • ERD5 protein, human
  • RNA, Messenger
  • Receptors, Estrogen
  • Progesterone
  • Estradiol