Phosphoproteomic analysis with a solid-phase capture-release-tag approach

Chem Biol. 2005 Jul;12(7):769-77. doi: 10.1016/j.chembiol.2005.05.012.

Abstract

A comprehensive study of global phosphorylation events in biological systems is critical. We report a chemistry-based capture-release-tag method for isolation of complex phospho-Ser/Thr-containing peptides by liquid beta-elimination combined with solid-phase Michael addition. The free thiol groups of 6-(mercapto-acetylamino)-hexanoic acid functionalized resin are used as immobilized Michael donors to capture dehydro-serine/threonine peptides. After an acid-mediated release step, phospho-peptides are labeled with a 6-(2-mercapto-acetylamine)-hexanoic amide tag at phosphorylated sites. We applied this method to analyze the phosphorylation status of microtubule-associated proteins. We find that a CDK5 substrate microtubule-associated protein 2 (MAP2) is phosphorylated on residues that are within a homologous region of Tau. The chemical method corroborates previous results and suggests that Tau and MAP2 may contain a CDK5 phosphorylation motif.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Binding Sites
  • Cyclin-Dependent Kinase 5
  • Cyclin-Dependent Kinases / metabolism
  • Cysteamine / chemistry
  • Isotope Labeling / methods*
  • Microtubule-Associated Proteins / analysis
  • Microtubule-Associated Proteins / chemistry
  • Molecular Sequence Data
  • Phosphoproteins / analysis*
  • Phosphoproteins / metabolism
  • Phosphorylation
  • Phosphoserine / analysis
  • Phosphoserine / chemistry
  • Phosphothreonine / chemistry
  • Phosphothreonine / metabolism
  • Proteomics / methods*
  • tau Proteins / chemistry
  • tau Proteins / metabolism

Substances

  • Microtubule-Associated Proteins
  • Phosphoproteins
  • tau Proteins
  • Phosphothreonine
  • Phosphoserine
  • Cysteamine
  • Cyclin-Dependent Kinase 5
  • Cyclin-Dependent Kinases