ICPBC and C12-ICPBC: two new red emitting, fluorescent Ca2+ indicators excited with visible light

Cell Calcium. 2006 Jan;39(1):3-11. doi: 10.1016/j.ceca.2005.09.003. Epub 2005 Oct 17.

Abstract

Two new, visible-excited and red-emitting fluorescent Ca(2+) indicators were synthesized and the spectral profiles of their free and Ca(2+) bound forms were studied. The fluorescent properties of these probes are due to the extended conjugation of the chromeno[3',2':3,4]pyrido[1,2a][1,3]benzimidazole chromophore incorporated in their BAPTA-type, Ca(2+) chelating structure. The compounds, namely ICPBC and its N-dodecyl analog C12-ICPBC exhibit Ca(2+) dissociation constants of 7.7 and 18.0 microM, respectively. The fluorescence spectra of the probes showed a clear shift in excitation wavelength maxima upon Ca(2+) binding along with a large Stokes shift and changes in fluorescence intensity, indicating their potential use as Ca(2+) indicators. The ability of ICPBC to trace high calcium spikes was tested in the human HepG2 cell line with positive results.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Algorithms
  • Benzimidazoles / chemical synthesis*
  • Benzimidazoles / chemistry
  • Benzopyrans / chemical synthesis*
  • Benzopyrans / chemistry
  • Calcium / analysis*
  • Cell Line
  • Fluorescent Dyes / chemical synthesis*
  • Fluorescent Dyes / chemistry
  • Humans
  • Indicators and Reagents / chemical synthesis
  • Indicators and Reagents / chemistry
  • Light*
  • Microscopy, Confocal / methods
  • Microscopy, Fluorescence

Substances

  • Benzimidazoles
  • Benzopyrans
  • C12-ICPBC compound
  • Fluorescent Dyes
  • ICPBC compound
  • Indicators and Reagents
  • Calcium