Okadaic acid inhibits activation of K-Cl cotransport in red blood cells containing hemoglobins S and C

Am J Physiol. 1991 Oct;261(4 Pt 1):C591-3. doi: 10.1152/ajpcell.1991.261.4.C591.

Abstract

The sensitivity of red blood cells containing hemoglobins S and C to activation of K-Cl cotransport by osmotic swelling and acidification was reduced by okadaic acid, a specific protein phosphatase inhibitor. The dose-response curve for okadaic acid suggests its action is on a type 1 protein phosphatase. Okadaic acid has been previously shown to inhibit swelling-induced activation of K-Cl cotransport in red blood cells from rabbits, normal humans, and dogs. The present work confirms the observation that okadaic acid blunts the stimulation of K-Cl cotransport by cell swelling. The new information is that okadaic acid reduces the effects of hemoglobins S and C on the volume and pH sensitivity of K-Cl cotransport. Thus the influences of cell volume, pH, and mutant hemoglobins may all be mediated via a common mechanisms that affects the phosphorylation state, either of the K-Cl. cotransporter itself or of a protein that regulates its function.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Carrier Proteins / blood*
  • Erythrocytes / metabolism*
  • Ethers, Cyclic / pharmacology*
  • Hemoglobin C / analysis*
  • Hemoglobin, Sickle / analysis*
  • Humans
  • Hydrogen-Ion Concentration
  • K Cl- Cotransporters
  • Okadaic Acid
  • Osmolar Concentration
  • Phosphoprotein Phosphatases / antagonists & inhibitors
  • Potassium / antagonists & inhibitors
  • Potassium / blood
  • Symporters*

Substances

  • Carrier Proteins
  • Ethers, Cyclic
  • Hemoglobin, Sickle
  • Symporters
  • Okadaic Acid
  • Hemoglobin C
  • Phosphoprotein Phosphatases
  • Potassium