The genetic stability of a conditional live HIV-1 variant can be improved by mutations in the Tet-On regulatory system that restrain evolution

J Biol Chem. 2006 Jun 23;281(25):17084-17091. doi: 10.1074/jbc.M513400200. Epub 2006 Apr 20.

Abstract

Live attenuated human immunodeficiency virus type 1 (HIV-1) vaccines are considered unsafe because more quickly replicating pathogenic virus variants may evolve after vaccination. As an alternative vaccine approach, we have previously presented a doxycycline (dox)-dependent HIV-1 variant that was constructed by incorporating the tetracycline-inducible gene expression system (Tet-On system) into the viral genome. Replication of this HIV-rtTA variant is driven by the dox-inducible transcriptional activator rtTA and can be switched on and off at will. A large scale evolution study was performed to test the genetic stability of this conditional live vaccine candidate. In several long term cultures, we selected for HIV-rtTA variants that no longer required dox for replication. These evolved variants acquired a typical amino acid substitution either at position 19 or 37 in the rtTA protein. Both mutations caused rtTA activity and viral replication in the absence of dox. We designed a novel rtTA variant with a higher genetic barrier toward these undesired evolutionary routes. The corresponding HIV-rtTA variant did not lose dox control in long term cultures, demonstrating its improved genetic stability.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • AIDS Vaccines / chemistry
  • AIDS Vaccines / genetics*
  • Codon
  • Doxycycline / metabolism
  • Evolution, Molecular
  • Gene Expression Regulation, Viral
  • Genetic Variation*
  • HIV Infections / prevention & control*
  • HIV-1 / genetics*
  • HeLa Cells
  • Humans
  • Mutation*
  • Tetracycline / pharmacology
  • Vaccines, Attenuated*
  • Virus Replication

Substances

  • AIDS Vaccines
  • Codon
  • Vaccines, Attenuated
  • Tetracycline
  • Doxycycline