Distance changes at the regulatory and catalytic sites on Escherichia coli glutamine synthetase: a spin label study on the effect of substrate(s) binding

Biochim Biophys Acta. 1991 Mar 8;1077(1):91-8. doi: 10.1016/0167-4838(91)90530-d.

Abstract

A spin-labeled ATP analogue, 2,2,6,6-tetramethylpiperidine-1-oxyl adenosine triphosphatase (Tempo-ATP) is used to adenylate Escherichia coli glutamine synthetase (L-glutamine: ammonia ligase (ADP-forming), EC 6.3.1.2). The Tempo adenylylated glutamine synthetase (Tempo-GS) exhibits similar catalytic properties, pH profile and inhibitor susceptibility as those of glutamine synthetase adenylylated with normal ATP. Using the spin label on the enzyme as a probe and employing the spin-spin interactions between the label probe and paramagnetic Mn2+, the distances from the nitroxyl moiety of the covalently bound Tempo-AMP to the two Mn2+ binding sites, n1 and n2 were determined. The n1 site is the structural site and n2 is located at the catalytic site. The distances from Mn2+ at n1 and n2 sites to the nitroxyl radical are 19 and 16 A, respectively. Binding of the substrate, L-Glu, causes a protein conformational change which is reflected by the reduction of approximately 2 A for the n1 to Tempo-AMP distance and lengthening of approximately 2 A for the n2 to the Tempo-AMP distance. Addition of ATP to the Tempo-GS/L-Glu complex increases the distance between n1 and Tempo-AMP, and n2 and Tempo-AMP by 4 and 3 A, respectively.

MeSH terms

  • Adenosine Diphosphate / metabolism
  • Adenosine Triphosphate / analogs & derivatives*
  • Adenosine Triphosphate / metabolism
  • Binding Sites
  • Cyclic N-Oxides / metabolism*
  • Electron Spin Resonance Spectroscopy
  • Escherichia coli / enzymology*
  • Glutamate-Ammonia Ligase / chemistry
  • Glutamate-Ammonia Ligase / metabolism*
  • Kinetics
  • Magnetic Resonance Spectroscopy
  • Protein Conformation
  • Spectrometry, Fluorescence
  • Spectrophotometry, Ultraviolet
  • Spin Labels

Substances

  • Cyclic N-Oxides
  • Spin Labels
  • 6-(2,2,6,6-tetramethylpiperidine-1-oxyl)-adenosine triphosphate
  • Adenosine Diphosphate
  • Adenosine Triphosphate
  • Glutamate-Ammonia Ligase