Effect of chemotherapy on somatostatin receptor detection with octreotide scintigraphy in hormone-refractory prostate cancer patients

Anticancer Res. 2006 May-Jun;26(3B):2233-5.

Abstract

Background: Neuroendocrine cells have been found in all stages of prostate cancer. Neuroendocrine differentiation of prostate adenocarcinoma is a possible target for therapeutic strategies, such as administration of GH analogs (e.g., somatostatin), especially in patients with hormone-refractory prostate cancer (HRPC). The presence of receptors for these drugs in tumor cells and tissues is essential and is assessed with 111In-octreotide scintigraphy (Octreoscan). The relationship between these receptors and chemotherapy, the new standard therapy for HRPC, is unknown.

Patients and methods: 111In-octreotide scintigraphy was performed on 20 patients affected by HRPC, all with metastatic disease. Chemotherapy with a single agent was also administered to all patients.

Results: In 63% of the patients, all metastases were negative to Octreoscan. Several metastases were positive in 37% of patients only, compared to 94% previously described in a chemotherapy-naive population.

Conclusion: Chemotherapy seemed to reduce the cellular receptors for somatostatin analogs.

MeSH terms

  • Aged
  • Aged, 80 and over
  • Antineoplastic Agents, Phytogenic / therapeutic use
  • Bone Neoplasms / diagnostic imaging
  • Bone Neoplasms / secondary
  • Docetaxel
  • Humans
  • Indium Radioisotopes* / metabolism
  • Male
  • Middle Aged
  • Octreotide / analogs & derivatives*
  • Octreotide / metabolism
  • Pentetic Acid / analogs & derivatives*
  • Pentetic Acid / metabolism
  • Positron-Emission Tomography
  • Prostatic Neoplasms / diagnostic imaging*
  • Prostatic Neoplasms / drug therapy*
  • Prostatic Neoplasms / pathology
  • Radiopharmaceuticals / metabolism
  • Receptors, Somatostatin / metabolism*
  • Taxoids / therapeutic use
  • Vinblastine / analogs & derivatives
  • Vinblastine / therapeutic use
  • Vinorelbine

Substances

  • Antineoplastic Agents, Phytogenic
  • Indium Radioisotopes
  • Radiopharmaceuticals
  • Receptors, Somatostatin
  • Taxoids
  • SDZ 215-811
  • Docetaxel
  • Vinblastine
  • Pentetic Acid
  • Vinorelbine
  • Octreotide