CD47 is necessary for inhibition of nitric oxide-stimulated vascular cell responses by thrombospondin-1

J Biol Chem. 2006 Sep 8;281(36):26069-80. doi: 10.1074/jbc.M605040200. Epub 2006 Jul 11.

Abstract

CD36 is necessary for inhibition of some angiogenic responses by the matricellular glycoprotein thrombospondin-1 and is therefore assumed to be the receptor that mediates its anti-angiogenic activities. Although ligation of CD36 by antibodies, recombinant type 1 repeats of thrombospondin-1, or CD36-binding peptides was sufficient to inhibit nitric oxide (NO)-stimulated responses in both endothelial and vascular smooth muscle cells, picomolar concentrations of native thrombospondin-1 similarly inhibited NO signaling in vascular cells from wild-type and CD36-null mice. Ligation of the thrombospondin-1 receptor CD47 by recombinant C-terminal regions of thrombospondin-1, thrombospondin-1 peptides, or CD47 antibodies was also sufficient to inhibit NO-stimulated phenotypic responses and cGMP signaling in vascular cells. Thrombospondin-1 did not inhibit NO signaling in CD47-null vascular cells or NO-stimulated vascular outgrowth from CD47-null muscle explants in three-dimensional cultures. Furthermore, the CD36-binding domain of thrombospondin-1 and anti-angiogenic peptides derived from this domain failed to inhibit NO signaling in CD47-null cells. Therefore, ligation of either CD36 or CD47 is sufficient to inhibit NO-stimulated vascular cell responses and cGMP signaling, but only CD47 is necessary for this activity of thrombospondin-1 at physiological concentrations.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, N.I.H., Intramural

MeSH terms

  • Animals
  • CD36 Antigens / genetics
  • CD36 Antigens / metabolism
  • CD47 Antigen / genetics
  • CD47 Antigen / metabolism*
  • Cell Adhesion / physiology
  • Cell Proliferation
  • Cells, Cultured
  • Cyclic GMP / metabolism
  • Endothelial Cells / cytology
  • Endothelial Cells / metabolism*
  • Humans
  • In Vitro Techniques
  • Ligands
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Muscle, Smooth, Vascular* / cytology
  • Muscle, Smooth, Vascular* / metabolism
  • Neovascularization, Physiologic
  • Nitric Oxide* / antagonists & inhibitors
  • Nitric Oxide* / metabolism
  • Peptides / genetics
  • Peptides / metabolism
  • Signal Transduction / physiology*
  • Thrombospondin 1 / metabolism*

Substances

  • CD36 Antigens
  • CD47 Antigen
  • Ligands
  • Peptides
  • Thrombospondin 1
  • Nitric Oxide
  • Cyclic GMP